Synthesis of glucosylated 1,2,3-triazole derivatives

被引：39

作者：

Chen, XM ^{[1
]}

Li, ZJ ^{[1
]}

Ren, ZX ^{[1
]}

Huang, ZT ^{[1
]}

机构：

[1] Chinese Acad Sci, Inst Chem, Beijing 100080, Peoples R China

来源：

CARBOHYDRATE RESEARCH | 1999年 / 315卷 / 3-4期

基金：

中国国家自然科学基金;

关键词：

synthesis; heterocycle; glucosylated; triazole;

D O I：

10.1016/S0008-6215(99)00020-8

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 [生物化学与分子生物学]; 081704 [应用化学];

摘要：

A series of potential bioactive compounds, l-glucosyl-4-heterocyclyl-5-(p-substituted-phenyl)-1,2,3-triazoles, were synthesized. Highly stereoselective products were obtained in good yield. Primary activity screening showed that this type of N-glucosylic compound possessed antitumour and antiviral activities. (C) 1999 Elsevier Science Ltd. All rights reserved.

引用

页码：262 / 267

页数：6

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