Deacetylase enzymes: biological functions and the use of small-molecule inhibitors

被引:490
作者
Grozinger, CM
Schreiber, SL
机构
[1] Harvard Univ, Dept Chem & Chem Biol, Cambridge, MA 02138 USA
[2] Harvard Univ, Howard Hughes Med Inst, Cambridge, MA 02138 USA
来源
CHEMISTRY & BIOLOGY | 2002年 / 9卷 / 01期
关键词
D O I
10.1016/S1074-5521(02)00092-3
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
[No abstract available]
引用
收藏
页码:3 / 16
页数:14
相关论文
共 100 条
[1]  
Aasland R, 1996, TRENDS BIOCHEM SCI, V21, P87, DOI 10.1016/0968-0004(96)30009-1
[2]   Characterization of a human gene with sequence homology to Saccharomyces cerevisiae SIR2 [J].
Afshar, G ;
Murnane, JP .
GENE, 1999, 234 (01) :161-168
[3]  
ALLFREY VG, 1971, HISTONES NUCLEOHISTO, P241
[4]   CoREST:: A functional corepressor required for regulation of neural-specific gene expression [J].
Andrés, ME ;
Burger, C ;
Peral-Rubio, MJ ;
Battaglioli, E ;
Anderson, ME ;
Grimes, J ;
Dallman, J ;
Ballas, N ;
Mandel, G .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1999, 96 (17) :9873-9878
[5]   Histone deacetylases: transcriptional repression with SINers and NuRDs [J].
Ayer, DE .
TRENDS IN CELL BIOLOGY, 1999, 9 (05) :193-198
[6]   THE SIR2 GENE FAMILY, CONSERVED FROM BACTERIA TO HUMANS, FUNCTIONS IN SILENCING, CELL-CYCLE PROGRESSION, AND CHROMOSOME STABILITY [J].
BRACHMANN, CB ;
SHERMAN, JM ;
DEVINE, SE ;
CAMERON, EE ;
PILLUS, L ;
BOEKE, JD .
GENES & DEVELOPMENT, 1995, 9 (23) :2888-2902
[7]  
Braunstein M, 1996, MOL CELL BIOL, V16, P4349
[8]   TRANSCRIPTIONAL SILENCING IN YEAST IS ASSOCIATED WITH REDUCED NUCLEOSOME ACETYLATION [J].
BRAUNSTEIN, M ;
ROSE, AB ;
HOLMES, SG ;
ALLIS, CD ;
BROACH, JR .
GENES & DEVELOPMENT, 1993, 7 (04) :592-604
[9]   Transcriptional silencing of Ty1 elements in the RDN1 locus of yeast [J].
Bryk, M ;
Banerjee, M ;
Murphy, M ;
Knudsen, KE ;
Garfinkel, DJ ;
Curcio, MJ .
GENES & DEVELOPMENT, 1997, 11 (02) :255-269
[10]   Co-repressors 2000 [J].
Burke, LJ ;
Baniahmad, A .
FASEB JOURNAL, 2000, 14 (13) :1876-1888