Convenient synthesis and transformation of 2,6-dichloro-4-iodopyridine

被引:34
作者
Mello, JV [1 ]
Finney, NS [1 ]
机构
[1] Univ Calif San Diego, Dept Chem & Biochem, La Jolla, CA 92093 USA
关键词
D O I
10.1021/ol0169269
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
[GRAPHICS] We describe a convenient scalable synthesis of 2,6-dichloro-4-iodopyridine and demonstrate its utility by stepwise elaboration to a number of 2,4,6-trisubstituted pyridines.
引用
收藏
页码:4263 / 4265
页数:3
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