One-pot preparation of 1-substituted imidazole-2-thione from isothiocyanate and amino acetal

被引：43

作者：

Matsuda, K

Yanagisawa, I

Isomura, Y

Mase, T

Shibanuma, T

机构：

[1] Inst. for Drug Discovery Research, Yamanouchi Pharmaceutical Co. Ltd., 21 Miyukigaoka, Tsukuba, Ibaraki

来源：

SYNTHETIC COMMUNICATIONS | 1997年 / 27卷 / 20期

关键词：

D O I：

10.1080/00397919708007078

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Isothiocyanates were treated with amino acetal and conc. HCl (0.5 eq.) successively in one-pot to afford 1-substituted imidazole-2-thiones in good yields.

引用

页码：3565 / 3571

页数：7

共 7 条

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