Synthesis of the first tricomponent bisubstrate analogue that exhibits potent inhibition against GlcNAc:beta-1,4-galactosyltransferase

被引：52

作者：

Hashimoto, H

Endo, T

Kajihara, Y

机构：

[1] Department of Life Science, Fac. of Bioscience and Biotechnology, Tokyo Institute of Technology, Midori-ku, Yokohama 226

[2] Nippon Chemipha Co., Misato 341

[3] Department of System Function, Yokohama City University, Kanazawa-ku, Yokohama 236, 22-6, Seto

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1997年 / 62卷 / 07期

关键词：

D O I：

10.1021/jo962235s

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[No abstract available]

引用

页码：1914 / 1915

页数：2

共 28 条

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[3] GLYCOPROTEIN BIOSYNTHESIS - STUDIES ON RECEPTOR SPECIFICITY OF POLYPEPTIDYL - N-ACETYLGALACTOSAMINYL TRANSFERASE FROM BOVINE SUBMAXIALLARY GLANDS
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[7] METHYL-3-O-(2-ACETAMIDO-2-DEOXY-6-THIO-BETA-D-GLUCOPYRANOSYL)-BETA-D-GALACTOPYRANOSIDE - A SLOW REACTING ACCEPTOR-ANALOG WHICH INHIBITS GLYCOSYLATION BY UDP-D-GALACTOSE-N-ACETYL-D-GLUCOSAMINE-(1-]4)-BETA-D-GALACTOSYLTRANSFERASE
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[J]. CARBOHYDRATE RESEARCH, 1992, 229 (01) : C5 - C9
[8] Kirby AJ, 1996, ANGEW CHEM INT EDIT, V35, P707
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[10] Lowe J B, 1991, Semin Cell Biol, V2, P289

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