共 10 条
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CNS and cutaneous involvement in patients with chronic myeloid leukemia treated with imatinib in hematologic complete remission: Two case reports
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Abruzzese, E
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Cantonetti, M
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Morino, L
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Orlandi, G
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Tendas, A
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Del Principe, MI
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Masi, M
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Amadori, S
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Orlandi, A
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Anemona, L
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Campione, E
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JOURNAL OF CLINICAL ONCOLOGY,
2003, 21 (22)
:4256-4258

Abruzzese, E
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Roma Tor Vergata, Dept Hematol, S Eugenio Hosp, Rome, Italy Univ Roma Tor Vergata, Dept Hematol, S Eugenio Hosp, Rome, Italy

Cantonetti, M
论文数: 0 引用数: 0
h-index: 0
机构: Univ Roma Tor Vergata, Dept Hematol, S Eugenio Hosp, Rome, Italy

Morino, L
论文数: 0 引用数: 0
h-index: 0
机构: Univ Roma Tor Vergata, Dept Hematol, S Eugenio Hosp, Rome, Italy

Orlandi, G
论文数: 0 引用数: 0
h-index: 0
机构: Univ Roma Tor Vergata, Dept Hematol, S Eugenio Hosp, Rome, Italy

Tendas, A
论文数: 0 引用数: 0
h-index: 0
机构: Univ Roma Tor Vergata, Dept Hematol, S Eugenio Hosp, Rome, Italy

Del Principe, MI
论文数: 0 引用数: 0
h-index: 0
机构: Univ Roma Tor Vergata, Dept Hematol, S Eugenio Hosp, Rome, Italy

Masi, M
论文数: 0 引用数: 0
h-index: 0
机构: Univ Roma Tor Vergata, Dept Hematol, S Eugenio Hosp, Rome, Italy

Amadori, S
论文数: 0 引用数: 0
h-index: 0
机构: Univ Roma Tor Vergata, Dept Hematol, S Eugenio Hosp, Rome, Italy

Orlandi, A
论文数: 0 引用数: 0
h-index: 0
机构: Univ Roma Tor Vergata, Dept Hematol, S Eugenio Hosp, Rome, Italy

Anemona, L
论文数: 0 引用数: 0
h-index: 0
机构: Univ Roma Tor Vergata, Dept Hematol, S Eugenio Hosp, Rome, Italy

Campione, E
论文数: 0 引用数: 0
h-index: 0
机构: Univ Roma Tor Vergata, Dept Hematol, S Eugenio Hosp, Rome, Italy
[2]
Breccia Massimo, 2004, Haematologica, V89, pECR11
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Comparative analysis of two clinically active BCR-ABL kinase inhibitors reveals the role of conformation-specific binding in resistance
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Skaggs, BJ
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Shah, NP
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Lee, FY
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Sawyers, CL
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PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
2005, 102 (09)
:3395-3400

Burgess, MR
论文数: 0 引用数: 0
h-index: 0
机构: Univ Calif Los Angeles, Div Hematol & Oncol, David Geffen Sch Med, Dept Med, Los Angeles, CA 90095 USA

Skaggs, BJ
论文数: 0 引用数: 0
h-index: 0
机构: Univ Calif Los Angeles, Div Hematol & Oncol, David Geffen Sch Med, Dept Med, Los Angeles, CA 90095 USA

Shah, NP
论文数: 0 引用数: 0
h-index: 0
机构: Univ Calif Los Angeles, Div Hematol & Oncol, David Geffen Sch Med, Dept Med, Los Angeles, CA 90095 USA

Lee, FY
论文数: 0 引用数: 0
h-index: 0
机构: Univ Calif Los Angeles, Div Hematol & Oncol, David Geffen Sch Med, Dept Med, Los Angeles, CA 90095 USA

Sawyers, CL
论文数: 0 引用数: 0
h-index: 0
机构: Univ Calif Los Angeles, Div Hematol & Oncol, David Geffen Sch Med, Dept Med, Los Angeles, CA 90095 USA
[4]
Imatinib mesylate resistance through BCR-ABL independence in chronic myelogenous leukemia
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Donato, NJ
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Wu, JY
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Stapley, J
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Lin, H
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Arlinghaus, R
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Aggarwal, B
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Shishodin, S
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Albitar, M
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Hayes, K
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Kantarjian, H
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Talpaz, M
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CANCER RESEARCH,
2004, 64 (02)
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Donato, NJ
论文数: 0 引用数: 0
h-index: 0
机构: Univ Texas, MD Anderson Canc Ctr, Dept Bioimmunotherapy, Houston, TX 77030 USA

Wu, JY
论文数: 0 引用数: 0
h-index: 0
机构: Univ Texas, MD Anderson Canc Ctr, Dept Bioimmunotherapy, Houston, TX 77030 USA

Stapley, J
论文数: 0 引用数: 0
h-index: 0
机构: Univ Texas, MD Anderson Canc Ctr, Dept Bioimmunotherapy, Houston, TX 77030 USA

Lin, H
论文数: 0 引用数: 0
h-index: 0
机构: Univ Texas, MD Anderson Canc Ctr, Dept Bioimmunotherapy, Houston, TX 77030 USA

Arlinghaus, R
论文数: 0 引用数: 0
h-index: 0
机构: Univ Texas, MD Anderson Canc Ctr, Dept Bioimmunotherapy, Houston, TX 77030 USA

Aggarwal, B
论文数: 0 引用数: 0
h-index: 0
机构: Univ Texas, MD Anderson Canc Ctr, Dept Bioimmunotherapy, Houston, TX 77030 USA

Shishodin, S
论文数: 0 引用数: 0
h-index: 0
机构: Univ Texas, MD Anderson Canc Ctr, Dept Bioimmunotherapy, Houston, TX 77030 USA

Albitar, M
论文数: 0 引用数: 0
h-index: 0
机构: Univ Texas, MD Anderson Canc Ctr, Dept Bioimmunotherapy, Houston, TX 77030 USA

Hayes, K
论文数: 0 引用数: 0
h-index: 0
机构: Univ Texas, MD Anderson Canc Ctr, Dept Bioimmunotherapy, Houston, TX 77030 USA

Kantarjian, H
论文数: 0 引用数: 0
h-index: 0
机构: Univ Texas, MD Anderson Canc Ctr, Dept Bioimmunotherapy, Houston, TX 77030 USA

Talpaz, M
论文数: 0 引用数: 0
h-index: 0
机构: Univ Texas, MD Anderson Canc Ctr, Dept Bioimmunotherapy, Houston, TX 77030 USA
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Discovery of N-(2-chloro-6-methylphenyl)-2-(6-(4-(2-hydroxyethyl)-piperazin-1-yl)-2-methylpyrimidin-4-ylamino)thiazole-5-carboxamide (BMS-354825), a dual Src/Abl kinase inhibitor with potent antitumor activity in preclinical assays
[J].
Lombardo, LJ
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Lee, FY
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Chen, P
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Norris, D
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Barrish, JC
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Behnia, K
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Castaneda, S
;
Cornelius, LAM
;
Das, J
;
Doweyko, AM
;
Fairchild, C
;
Hunt, JT
;
Inigo, I
;
Johnston, K
;
Kamath, A
;
Kan, D
;
Klei, H
;
Marathe, P
;
Pang, SH
;
Peterson, R
;
Pitt, S
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Schieven, GL
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Schmidt, RJ
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Tokarski, J
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Wen, ML
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Wityak, J
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Borzilleri, RM
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JOURNAL OF MEDICINAL CHEMISTRY,
2004, 47 (27)
:6658-6661

Lombardo, LJ
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Lee, FY
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Chen, P
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Norris, D
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Barrish, JC
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Behnia, K
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Castaneda, S
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Cornelius, LAM
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Das, J
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Doweyko, AM
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Fairchild, C
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Hunt, JT
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Inigo, I
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Johnston, K
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Kamath, A
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Kan, D
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Klei, H
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Marathe, P
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Pang, SH
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Peterson, R
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Pitt, S
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Schieven, GL
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Schmidt, RJ
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Tokarski, J
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Wen, ML
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Wityak, J
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA

Borzilleri, RM
论文数: 0 引用数: 0
h-index: 0
机构:
Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Pharmaceut Res Inst, Princeton, NJ 08543 USA
[7]
In vitro activity of Bcr-Abl inhibitors AMN107 and BMS-354825 against clinically relevant imatinib-resistant Abl kinase domain mutants
[J].
O'Hare, T
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Walters, DK
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Stoffregen, EP
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Jia, TP
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Manley, PW
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Mestan, J
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Cowan-Jacob, SW
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Lee, FY
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Heinrich, MC
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Deininger, MWN
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Druker, BJ
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CANCER RESEARCH,
2005, 65 (11)
:4500-4505

O'Hare, T
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Walters, DK
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Stoffregen, EP
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Jia, TP
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Manley, PW
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Mestan, J
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Cowan-Jacob, SW
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Lee, FY
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Heinrich, MC
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Deininger, MWN
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Druker, BJ
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA
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Overriding imatinib resistance with a novel ABL kinase inhibitor
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Shah, NP
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SCIENCE,
2004, 305 (5682)
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Shah, NP
论文数: 0 引用数: 0
h-index: 0
机构: Univ Calif Los Angeles, Dept Med, Div Hematol & Oncol, Los Angeles, CA 90095 USA

Tran, C
论文数: 0 引用数: 0
h-index: 0
机构: Univ Calif Los Angeles, Dept Med, Div Hematol & Oncol, Los Angeles, CA 90095 USA

Lee, FY
论文数: 0 引用数: 0
h-index: 0
机构: Univ Calif Los Angeles, Dept Med, Div Hematol & Oncol, Los Angeles, CA 90095 USA

Chen, P
论文数: 0 引用数: 0
h-index: 0
机构: Univ Calif Los Angeles, Dept Med, Div Hematol & Oncol, Los Angeles, CA 90095 USA

Norris, D
论文数: 0 引用数: 0
h-index: 0
机构: Univ Calif Los Angeles, Dept Med, Div Hematol & Oncol, Los Angeles, CA 90095 USA

Sawyers, CL
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif Los Angeles, Dept Med, Div Hematol & Oncol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Med, Div Hematol & Oncol, Los Angeles, CA 90095 USA
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ABL mutations in late chronic phase chronic myeloid leukemia patients with up-front cytogenetic resistance to imatinib are associated with a greater likelihood of progression to blast crisis and shorter survival: A study by the GIMEMA working party on chronic myeloid leukemia
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Soverini, S
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Martinelli, G
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Trabacchi, E
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Castagnetti, F
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Testoni, N
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Luatti, S
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de Vivo, A
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Cilloni, D
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Izzo, B
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Fava, M
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Abruzzese, E
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Pane, F
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JOURNAL OF CLINICAL ONCOLOGY,
2005, 23 (18)
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Soverini, S
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Martinelli, G
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Rosti, G
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Bassi, S
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Amabile, M
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Poerio, A
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Giannini, B
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Trabacchi, E
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Castagnetti, F
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Testoni, N
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Luatti, S
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

de Vivo, A
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Cilloni, D
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Izzo, B
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Fava, M
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Abruzzese, E
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Alberti, D
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Pane, F
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Saglio, G
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy

Baccarani, M
论文数: 0 引用数: 0
h-index: 0
机构: Univ Bologna, Inst Hematol & Med Oncol Seragnoli, I-40138 Bologna, Italy
