Semisynthesis of 3-β-hydroxyartemisinin

被引：6

作者：

Acton, N ^{[1
]}

机构：

[1] Walter Reed Army Med Ctr, Walter Reed Army Inst Res, Div Expt Therapeut, Washington, DC 20307 USA

来源：

JOURNAL OF NATURAL PRODUCTS | 1999年 / 62卷 / 05期

关键词：

D O I：

10.1021/np980555w

中图分类号：

Q94 [植物学];

学科分类号：

071001 ;

摘要：

3-beta-Hydroxyartemisinin (5) was synthesized from 3-beta-hydroxydihydroartemisinic acid (7c) via singlet oxygen oxidation followed by air (triplet oxygen) oxidation. Compound 7c was synthesized in two steps from dihydroartemisinic acid, 7a.

引用

页码：790 / 793

页数：4

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