In vitro photo-release of a TRPV1 agonist

被引:18
作者
Carr, JL
Wease, KN
Van Ryssen, MP
Paterson, S
Agate, B
Gallagher, KA
Brown, CTA
Scott, RH
Conway, SJ [1 ]
机构
[1] Univ St Andrews, EaStCHEM, Sch Chem, St Andrews KY16 9ST, Fife, Scotland
[2] Univ St Andrews, Ctr Biomol Sci, St Andrews KY16 9ST, Fife, Scotland
[3] Univ St Andrews, Sch Phys & Astron, St Andrews KY16 9ST, Fife, Scotland
[4] Univ Aberdeen, Inst Med Sci, Aberdeen AB25 2ZD, Scotland
关键词
D O I
10.1016/j.bmcl.2005.09.018
中图分类号
R914 [药物化学];
学科分类号
100701 [药物化学];
摘要
Intracellular photolysis of a novel 'caged' capsaicin analogue results in in vitro activation of the capsaicin receptor TRPV1. (c) 2005 Elsevier Ltd. All rights reserved.
引用
收藏
页码:208 / 212
页数:5
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