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Regiochemistry in Stille couplings of 2,6-dihalopurines

被引：92
作者：
Langli, G
Gundersen, LL
Rise, F
机构：
[1] OSLO COLL,DEPT HLTH,PROGRAM PHARM,N-0167 OSLO,NORWAY
[2] UNIV OSLO,DEPT CHEM,N-0315 OSLO,NORWAY
来源：
TETRAHEDRON | 1996年 / 52卷 / 15期
关键词：
D O I：
10.1016/0040-4020(96)00199-8
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The regiochemistry in Stille couplings of 2,6-dihalopurines have been studied. 2,6-Dichloropurines react selectively in the B-position, and 6-chloro-2-iodopurines and 2-bromo-6-chloropurines in the 3-position. Copyright (C) 1996 Elsevier Science Ltd
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页码：5625 / 5638
页数：14
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