Novel fluoroketolides: synthesis and antibacterial activity

被引:7
作者
Denis, A
Bonnefoy, A
机构
[1] Aventis Pharma, Med Chem, F-93235 Romainville, France
[2] Aventis Pharma, Infect Dis Grp 102, F-93235 Romainville, France
关键词
D O I
10.1358/dof.2001.026.10.633694
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
[No abstract available]
引用
收藏
页码:975 / 984
页数:10
相关论文
共 29 条
[1]   Synthesis and antibacterial activity of ketolides (6-O-methyl-3-oxoerythromycin derivatives):: A new class of antibacterials highly potent against macrolide-resistant and -susceptible respiratory pathogens [J].
Agouridas, C ;
Denis, A ;
Auger, JM ;
Benedetti, Y ;
Bonnefoy, A ;
Bretin, F ;
Chantot, JF ;
Dussarat, A ;
Fromentin, C ;
D'Ambrières, SG ;
Lachaud, S ;
Laurin, P ;
Le Martret, O ;
Loyau, V ;
Tessot, N .
JOURNAL OF MEDICINAL CHEMISTRY, 1998, 41 (21) :4080-4100
[2]  
AGOURIDAS C, 1997, 37 INT C ANT AG CHEM
[3]  
AGOURIDAS C, Patent No. 2742757
[4]  
AGOURIDAS C, 1998, INT C MACR AZ STREPT
[5]  
AGOURIDAS C, Patent No. 2785612
[6]   Ketolides lack inducibility properties of MLSB resistance phenotype [J].
Bonnefoy, A ;
Girard, AM ;
Agouridas, C ;
Chantot, JF .
JOURNAL OF ANTIMICROBIAL CHEMOTHERAPY, 1997, 40 (01) :85-90
[7]  
BONNEFOY A, 1999, 39 INT C ANT AG CHEM
[8]   The in-vitro activity of HMR 3647, a new ketolide antimicrobial agent [J].
Boswell, FJ ;
Andrews, JM ;
Ashby, JP ;
Fogarty, C ;
Brenwald, NP ;
Wise, R .
JOURNAL OF ANTIMICROBIAL CHEMOTHERAPY, 1998, 42 (06) :703-709
[9]  
CHU D, Patent No. 0063224
[10]   β-keto-ester chemistry and ketolides.: Synthesis and antibacterial activity of 2-halogeno, 2-methyl and 2,3 enol-ether ketolides [J].
Denis, A ;
Bretin, F ;
Fromentin, C ;
Bonnet, A ;
Piltan, G ;
Bonnefoy, A ;
Agouridas, C .
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2000, 10 (17) :2019-2022