Chemoselective three-component coupling via a tandem Pd-catalyzed boron-Heck and Suzuki reactions

被引：10

作者：

O'Neill, Justin

Yoo, Kyung Soo

Jung, Kyung Woon ^{[1
]}

机构：

[1] Univ So Calif, Loker Hydrocarbon Res Inst, Los Angeles, CA 90089 USA

来源：

TETRAHEDRON LETTERS | 2008年 / 49卷 / 51期

基金：

美国国家卫生研究院;

关键词：

D O I：

10.1016/j.tetlet.2008.10.039

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A new approach is herein reported to prepare biaryl derivatives via a tandem Pd-catalyzed boron-Heck and Suzuki reactions. This one-pot tandem process avoided purification or addition of extra catalyst between steps. The resulting biaryl compounds can be prepared with substrate variability in good to moderate yields. (C) 2008 Elsevier Ltd. All rights reserved.

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收藏

页码：7307 / 7310

页数：4

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