HIV-1 entry inhibitors in the side pocket

被引:84
作者
Sodroski, JG [1 ]
机构
[1] Harvard Univ, Sch Med, Dept Canc Immunol & AIDS, Boston, MA 02115 USA
[2] Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA
[3] Harvard Univ, Sch Med, Dept Pathol, Boston, MA 02115 USA
[4] Harvard Univ, Sch Publ Hlth, Dept Immunol & Infect Dis, Boston, MA 02115 USA
关键词
D O I
10.1016/S0092-8674(00)81655-4
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
[No abstract available]
引用
收藏
页码:243 / 246
页数:4
相关论文
共 18 条
  • [1] EFFECTS OF AMINO-ACID CHANGES IN THE EXTRACELLULAR DOMAIN OF THE HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 GP41 ENVELOPE GLYCOPROTEIN
    CAO, J
    BERGERON, L
    HELSETH, E
    THALI, M
    REPKE, H
    SODROSKI, J
    [J]. JOURNAL OF VIROLOGY, 1993, 67 (05) : 2747 - 2755
  • [2] Core structure of gp41 from the HIV envelope glycoprotein
    Chan, DC
    Fass, D
    Berger, JM
    Kim, PS
    [J]. CELL, 1997, 89 (02) : 263 - 273
  • [3] Evidence that a prominent cavity in the coiled coil of HIV type 1 gp41 is an attractive drug target
    Chan, DC
    Chutkowski, CT
    Kim, PS
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1998, 95 (26) : 15613 - 15617
  • [4] HIV entry and its inhibition
    Chan, DC
    Kim, PS
    [J]. CELL, 1998, 93 (05) : 681 - 684
  • [5] MUTATIONS IN THE LEUCINE ZIPPER OF THE HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 TRANSMEMBRANE GLYCOPROTEIN AFFECT FUSION AND INFECTIVITY
    DUBAY, JW
    ROBERTS, SJ
    BRODY, B
    HUNTER, E
    [J]. JOURNAL OF VIROLOGY, 1992, 66 (08) : 4748 - 4756
  • [6] Inhibiting HIV-1 entry: Discovery of D-peptide inhibitors that target the gp41 coiled-coil pocket
    Eckert, DM
    Malashkevich, VN
    Hong, LH
    Carr, PA
    Kim, PS
    [J]. CELL, 1999, 99 (01) : 103 - 115
  • [7] Ferrer M, 1999, NAT STRUCT BIOL, V6, P953
  • [8] Capture of an early fusion-active conformation of HIV-1 gp41
    Furuta, RA
    Wild, CT
    Weng, YK
    Weiss, CD
    [J]. NATURE STRUCTURAL BIOLOGY, 1998, 5 (04) : 276 - 279
  • [9] HIV-1 INHIBITION BY A PEPTIDE
    JIANG, SB
    LIN, K
    STRICK, N
    NEURATH, AR
    [J]. NATURE, 1993, 365 (6442) : 113 - 113
  • [10] Potent suppression of HIV-1 replication in humans by T-20, a peptide inhibitor of gp41-mediated virus entry
    Kilby, JM
    Hopkins, S
    Venetta, TM
    DiMassimo, B
    Cloud, GA
    Lee, JY
    Alldredge, L
    Hunter, E
    Lambert, D
    Bolognesi, D
    Mathews, T
    Johnson, MR
    Nowak, MA
    Shaw, GM
    Saag, MS
    [J]. NATURE MEDICINE, 1998, 4 (11) : 1302 - 1307