Parallel kinetic resolution of racemic amines using 3-N,N-diacylaminoquinazolin-4(3H)-ones

被引：15

作者：

Al-Sehemi, AG ^{[1
]}

Atkinson, RS ^{[1
]}

Meades, CK ^{[1
]}

机构：

[1] Univ Leicester, Dept Chem, Leicester LE1 7RH, Leics, England

来源：

CHEMICAL COMMUNICATIONS | 2001年 / 24期

关键词：

D O I：

10.1039/b109297a

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

The two pseudoenantiotopic N-acyl groups of enantiopure 3-[N-(3-m-acetoxyphenylpropanoyl)-N-(3-phenylpropanoyl)amine]-2-isopropylquinazolin-4(3H)-one 7 each react with a different enantiomer of 2-methylpiperidine giving rise to efficient parallel kinetic resolution (ee > 95%).

引用

页码：2684 / 2685

页数：2

共 8 条

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