First total synthesis of Mer-N5075A, a new HIV-I protease inhibitor from Streptomyces chromofuscus

被引：4

作者：

Konda, Y ^{[1
]}

Takahashi, Y ^{[1
]}

Mita, H ^{[1
]}

Takeda, K ^{[1
]}

Harigaya, Y ^{[1
]}

机构：

[1] KITASATO UNIV, SCH SCI, DEPT CHEM, SAGAMIHARA, KANAGAWA 228, JAPAN

来源：

CHEMISTRY LETTERS | 1997年 / 04期

关键词：

D O I：

10.1246/cl.1997.345

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

The first total synthesis of Mer-N5075A (1), a new potential HIV-I protease inhibitor produced from,Streptomyces chromofuscus, was achieved. The synthetic method is available for Mer-N5075A analogues such as alpha-MAPI (2), GE20372 A (4) and other chemically modified compounds.

引用

页码：345 / 346

页数：2

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