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Characteristics and common properties of inhibitors, inducers, and activators of CYP enzymes
被引:171
作者
:
Hollenberg, PF
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Michigan, Ann Arbor, MI 48109 USA
Univ Michigan, Ann Arbor, MI 48109 USA
Hollenberg, PF
[
1
]
机构
:
[1]
Univ Michigan, Ann Arbor, MI 48109 USA
来源
:
DRUG METABOLISM REVIEWS
|
2002年
/ 34卷
/ 1-2期
关键词
:
D O I
:
10.1081/DMR-120001387
中图分类号
:
R9 [药学];
学科分类号
:
1007 ;
摘要
:
[No abstract available]
引用
收藏
页码:17 / 35
页数:19
相关论文
共 63 条
[1]
ACETONE ENHANCEMENT OF MICROSOMAL ANILINE PARA-HYDROXYLASE ACTIVITY
ANDERS, MW
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Physiology, Biochemistry and Pharmacology, New York Stale Veterinary College, Cornell University, Ithaca
ANDERS, MW
[J].
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS,
1968,
126
(01)
: 269
-
+
[2]
ANDERS MW, 1973, PROGR DRUG RES, V17, P11
[3]
Allosteric behavior in cytochrome P450-dependent in vitro drug-drug interactions: A prospective based on conformational dynamics
Atkins, WM
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Washington, Dept Med Chem, Seattle, WA 98195 USA
Univ Washington, Dept Med Chem, Seattle, WA 98195 USA
Atkins, WM
Wang, RW
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Washington, Dept Med Chem, Seattle, WA 98195 USA
Wang, RW
Lu, AYH
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Washington, Dept Med Chem, Seattle, WA 98195 USA
Lu, AYH
[J].
CHEMICAL RESEARCH IN TOXICOLOGY,
2001,
14
(04)
: 338
-
347
[4]
Ator M. A., 1990, ENZYMES, V19, P214
[5]
Rifampin drastically reduces plasma concentrations and effects of oral midazolam
Backman, JT
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Clinical Pharmacology, University of Helsinki
Backman, JT
Olkkola, KT
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Clinical Pharmacology, University of Helsinki
Olkkola, KT
Neuvonen, PJ
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Clinical Pharmacology, University of Helsinki
Neuvonen, PJ
[J].
CLINICAL PHARMACOLOGY & THERAPEUTICS,
1996,
59
(01)
: 7
-
13
[6]
OXIDATION OF BENZO[A]PYRENE BY RECOMBINANT HUMAN CYTOCHROME-P450 ENZYMES
BAUER, E
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
BAUER, E
GUO, ZY
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
GUO, ZY
UENG, YF
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
UENG, YF
BELL, LC
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
BELL, LC
ZELDIN, D
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
ZELDIN, D
GUENGERICH, FP
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
GUENGERICH, FP
[J].
CHEMICAL RESEARCH IN TOXICOLOGY,
1995,
8
(01)
: 136
-
142
[7]
Black DJ, 1996, DRUG METAB DISPOS, V24, P422
[8]
BOUCHER PD, 1995, MOL CELL BIOL, V15, P5144
[9]
IN-VITRO BINDING AND FUNCTIONAL-STUDIES COMPARING THE HUMAN CYP1A1 NEGATIVE REGULATORY ELEMENT WITH THE ORTHOLOGOUS SEQUENCES FROM RODENT GENES
BOUCHER, PD
论文数:
0
引用数:
0
h-index:
0
机构:
WAYNE STATE UNIV, SCH MED, DEPT PHARMACOL, DETROIT, MI 48201 USA
WAYNE STATE UNIV, SCH MED, DEPT PHARMACOL, DETROIT, MI 48201 USA
BOUCHER, PD
HINES, RN
论文数:
0
引用数:
0
h-index:
0
机构:
WAYNE STATE UNIV, SCH MED, DEPT PHARMACOL, DETROIT, MI 48201 USA
WAYNE STATE UNIV, SCH MED, DEPT PHARMACOL, DETROIT, MI 48201 USA
HINES, RN
[J].
CARCINOGENESIS,
1995,
16
(02)
: 383
-
392
[10]
VIRTUAL KINETICS - USING STATISTICAL EXPERIMENTAL-DESIGN FOR RAPID ANALYSIS OF ENZYME-INHIBITOR MECHANISMS
BRONSON, DD
论文数:
0
引用数:
0
h-index:
0
机构:
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
BRONSON, DD
DANIELS, DM
论文数:
0
引用数:
0
h-index:
0
机构:
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
DANIELS, DM
DIXON, JT
论文数:
0
引用数:
0
h-index:
0
机构:
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
DIXON, JT
REDICK, CC
论文数:
0
引用数:
0
h-index:
0
机构:
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
REDICK, CC
HAALAND, PD
论文数:
0
引用数:
0
h-index:
0
机构:
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
HAALAND, PD
[J].
BIOCHEMICAL PHARMACOLOGY,
1995,
50
(06)
: 823
-
831
←
1
2
3
4
5
6
7
→
共 63 条
[1]
ACETONE ENHANCEMENT OF MICROSOMAL ANILINE PARA-HYDROXYLASE ACTIVITY
ANDERS, MW
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Physiology, Biochemistry and Pharmacology, New York Stale Veterinary College, Cornell University, Ithaca
ANDERS, MW
[J].
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS,
1968,
126
(01)
: 269
-
+
[2]
ANDERS MW, 1973, PROGR DRUG RES, V17, P11
[3]
Allosteric behavior in cytochrome P450-dependent in vitro drug-drug interactions: A prospective based on conformational dynamics
Atkins, WM
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Washington, Dept Med Chem, Seattle, WA 98195 USA
Univ Washington, Dept Med Chem, Seattle, WA 98195 USA
Atkins, WM
Wang, RW
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Washington, Dept Med Chem, Seattle, WA 98195 USA
Wang, RW
Lu, AYH
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Washington, Dept Med Chem, Seattle, WA 98195 USA
Lu, AYH
[J].
CHEMICAL RESEARCH IN TOXICOLOGY,
2001,
14
(04)
: 338
-
347
[4]
Ator M. A., 1990, ENZYMES, V19, P214
[5]
Rifampin drastically reduces plasma concentrations and effects of oral midazolam
Backman, JT
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Clinical Pharmacology, University of Helsinki
Backman, JT
Olkkola, KT
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Clinical Pharmacology, University of Helsinki
Olkkola, KT
Neuvonen, PJ
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Clinical Pharmacology, University of Helsinki
Neuvonen, PJ
[J].
CLINICAL PHARMACOLOGY & THERAPEUTICS,
1996,
59
(01)
: 7
-
13
[6]
OXIDATION OF BENZO[A]PYRENE BY RECOMBINANT HUMAN CYTOCHROME-P450 ENZYMES
BAUER, E
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
BAUER, E
GUO, ZY
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
GUO, ZY
UENG, YF
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
UENG, YF
BELL, LC
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
BELL, LC
ZELDIN, D
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
ZELDIN, D
GUENGERICH, FP
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,SCH MED,DEPT BIOCHEM,NASHVILLE,TN 37232
GUENGERICH, FP
[J].
CHEMICAL RESEARCH IN TOXICOLOGY,
1995,
8
(01)
: 136
-
142
[7]
Black DJ, 1996, DRUG METAB DISPOS, V24, P422
[8]
BOUCHER PD, 1995, MOL CELL BIOL, V15, P5144
[9]
IN-VITRO BINDING AND FUNCTIONAL-STUDIES COMPARING THE HUMAN CYP1A1 NEGATIVE REGULATORY ELEMENT WITH THE ORTHOLOGOUS SEQUENCES FROM RODENT GENES
BOUCHER, PD
论文数:
0
引用数:
0
h-index:
0
机构:
WAYNE STATE UNIV, SCH MED, DEPT PHARMACOL, DETROIT, MI 48201 USA
WAYNE STATE UNIV, SCH MED, DEPT PHARMACOL, DETROIT, MI 48201 USA
BOUCHER, PD
HINES, RN
论文数:
0
引用数:
0
h-index:
0
机构:
WAYNE STATE UNIV, SCH MED, DEPT PHARMACOL, DETROIT, MI 48201 USA
WAYNE STATE UNIV, SCH MED, DEPT PHARMACOL, DETROIT, MI 48201 USA
HINES, RN
[J].
CARCINOGENESIS,
1995,
16
(02)
: 383
-
392
[10]
VIRTUAL KINETICS - USING STATISTICAL EXPERIMENTAL-DESIGN FOR RAPID ANALYSIS OF ENZYME-INHIBITOR MECHANISMS
BRONSON, DD
论文数:
0
引用数:
0
h-index:
0
机构:
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
BRONSON, DD
DANIELS, DM
论文数:
0
引用数:
0
h-index:
0
机构:
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
DANIELS, DM
DIXON, JT
论文数:
0
引用数:
0
h-index:
0
机构:
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
DIXON, JT
REDICK, CC
论文数:
0
引用数:
0
h-index:
0
机构:
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
REDICK, CC
HAALAND, PD
论文数:
0
引用数:
0
h-index:
0
机构:
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
BECTON DICKINSON RES CTR,RES TRIANGLE PK,NC 27709
HAALAND, PD
[J].
BIOCHEMICAL PHARMACOLOGY,
1995,
50
(06)
: 823
-
831
←
1
2
3
4
5
6
7
→