Metal ion-assisted peptide cyclization

被引：42

作者：

Zhang, LS ^{[1
]}

Tam, JP ^{[1
]}

机构：

[1] VANDERBILT UNIV,DEPT IMMUNOL & MICROBIOL,MED CTR N A5119,NASHVILLE,TN 37232

来源：

TETRAHEDRON LETTERS | 1997年 / 38卷 / 25期

关键词：

D O I：

10.1016/S0040-4039(97)00935-0

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

We describe an efficient chemoselective method for Ag+ ion-assisted lactamization or lactonization of linear peptides to obtain end-to-end and sidechain-to-end cyclic peptides in aqueous buffered solutions. (C) 1997 Elsevier Science Ltd.

引用

页码：4375 / 4378

页数：4

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