Synthesis of 6-allyl and 6-heteroarylindoles by palladium catalyzed Stille cross-coupling reaction

被引：19

作者：

Benhida, R ^{[1
]}

Lecubin, F

Fourrey, JL

Castellanos, LR

Quintero, L

机构：

[1] CNRS, Inst Chim Subst Nat, F-91198 Gif Sur Yvette, France

[2] Univ Autonoma Puebla, CIFQ, Puebla 72570, Mexico

来源：

TETRAHEDRON LETTERS | 1999年 / 40卷 / 31期

关键词：

heteroarylindoles; Stille cross-coupling; palladium catalysts;

D O I：

10.1016/S0040-4039(99)01094-1

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Several 6-allyl and 6-heteroarylindoles have been synthesized in high yield by means of palladium catalyzed cross-coupling reactions between tributyltin derivatives and 6-haloindoles to give useful intermediates for the synthesis of analogues of biologically active natural products. (C) 1999 Elsevier Science Ltd. All rights reserved.

引用

页码：5701 / 5703

页数：3

共 4 条

[1] Indole arylation studies directed towards the synthesis of simplified eastern subunits of chloropeptin and kistamycin
Carbonnelle, AC
Zamora, EG
Beugelmans, R
Roussi, G
[J]. TETRAHEDRON LETTERS, 1998, 39 (25) : 4467 - 4470
[2] Complestatin and chloropeptin I, condensed aromatic peptides from two strains of streptomycetes
Hegde, VR
Dai, P
Patel, M
Gullo, VP
[J]. TETRAHEDRON LETTERS, 1998, 39 (32) : 5683 - 5684
[3] THE PALLADIUM-CATALYZED CROSS-COUPLING REACTIONS OF ORGANOTIN REAGENTS WITH ORGANIC ELECTROPHILES
STILLE, JK
[J]. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH, 1986, 25 (06): : 508 - 523
[4] Recent progress in the chemistry of non-monoterpenoid indole alkaloids
Toyota, M
Ihara, N
[J]. NATURAL PRODUCT REPORTS, 1998, 15 (04) : 327 - 340

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