A simple synthesis of 2-substituted oxazolines and oxazines

被引：104

作者：

Cwik, A

Hell, Z ^{[1
]}

Hegedüs, A

Finta, Z

Horváth, Z

机构：

[1] Budapest Univ Technol & Econ, Dept Organ Chem Technol, H-1521 Budapest, Hungary

[2] Erdokemia Ker Ltd, H-1108 Budapest, Hungary

来源：

TETRAHEDRON LETTERS | 2002年 / 43卷 / 22期

基金：

匈牙利科学研究基金会;

关键词：

D O I：

10.1016/S0040-4039(02)00723-2

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

beta-Aminoalcohols react with carboxylic acids in the presence of a zeolite, Ersorb-4, resulting in the formation of oxazoline derivatives in good yields. Similarly, 3-aminopropanol and benzoic acid gave the corresponding 2-phenyloxazine. (C) 2002 Elsevier Science Ltd. All rights reserved.

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收藏

页码：3985 / 3987

页数：3

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