Regio- and selective synthesis of 4,6-disubstituted-2-pyridones

被引:26
作者
Cherry, K
Abarbri, M
Parrain, JL
Duchêne, A
机构
[1] Fac Sci Tours, Lab Physicochim Interfaces & Millieuz React, F-37200 Tours, France
[2] Fac Sci & Tech St Jerome, CNRS, UMR 6009, Organ Synth Lab, F-13397 Marseille 20, France
关键词
2-pyridones; tributylstannylallenes; palladium catalyst; coupling reactions;
D O I
10.1016/S0040-4039(03)01429-1
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Palladium catalysed regio- and stereoselective annulation of allenyl stannanes by beta-iodo vinylic arnides gives good yields of the corresponding 2-pyridones. This annulation probably occurs via a Stille reaction/cyclisation sequence. (C) 2003 Elsevier Ltd. All rights reserved.
引用
收藏
页码:5791 / 5794
页数:4
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