Conformationally constrained 1,3-diamino ketones: A series of potent inhibitors of the cysteine protease cathepsin K

被引：51

作者：

Marquis, RW

Yamashita, DS

Ru, Y

LoCastro, SM

Oh, HJ

Erhard, KF

DesJarlais, RL

Head, MS

Smith, WW

Zhao, BG

Janson, CA

Abdel-Meguid, SS

Tomaszek, TA

Levy, MA

Veber, DF

机构：

[1] SmithKline Beecham Pharmaceut, Dept Med Chem, King Of Prussia, PA 19406 USA

[2] SmithKline Beecham Pharmaceut, Dept Phys & Struct Chem, King Of Prussia, PA 19406 USA

[3] SmithKline Beecham Pharmaceut, Dept Biol Struct, King Of Prussia, PA 19406 USA

[4] SmithKline Beecham Pharmaceut, Dept Mol Recognit, King Of Prussia, PA 19406 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1998年 / 41卷 / 19期

关键词：

D O I：

10.1021/jm980295f

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：3563 / 3567

页数：5

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