Iontophoresis of nafarelin across human skin in vitro

被引:13
作者
Bayon, AMR
Guy, RH
机构
[1] UNIV CALIF SAN FRANCISCO, DEPT BIOPHARMACEUT SCI, SAN FRANCISCO, CA 94143 USA
[2] UNIV CALIF SAN FRANCISCO, DEPT PHARMACEUT CHEM, SAN FRANCISCO, CA 94143 USA
[3] UNIV COMPLUTENSE MADRID, FAC FARM, DEPT FARM & TECNOL FARMACEUT, E-28040 MADRID, SPAIN
关键词
iontophoresis; electroosmosis; nafarelin; transdermal drug delivery; peptides;
D O I
10.1023/A:1016072205371
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
[No abstract available]
引用
收藏
页码:798 / 800
页数:3
相关论文
共 19 条
[1]  
BAYON AMR, 1994, P INT S CONTR REL BI, V21, P375
[2]  
BURNETTE RR, 1989, TRANSDERMAL DRUG DEL, P247
[3]   ABSORPTION AND METABOLISM OF NAFARELIN, A POTENT AGONIST OF GONADOTROPIN-RELEASING HORMONE [J].
CHAN, RL ;
HENZL, MR ;
LEPAGE, ME ;
LAFARGUE, J ;
NERENBERG, CA ;
ANIK, S ;
CHAPLIN, MD .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1988, 44 (03) :275-282
[4]   PENETRATION ENHANCEMENT FOR POLYPEPTIDES THROUGH EPITHELIA .D. ROUTES OF DELIVERY - CASE-STUDIES .6. TRANSDERMAL DELIVERY OF PEPTIDES AND PROTEINS [J].
CULLANDER, C ;
GUY, RH .
ADVANCED DRUG DELIVERY REVIEWS, 1992, 8 (2-3) :291-329
[5]   IONTOPHORETIC DELIVERY OF NAFARELIN ACROSS THE SKIN [J].
DELGADOCHARRO, MB ;
GUY, RH .
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 1995, 117 (02) :165-172
[6]   IONTOPHORESIS OF NAFARELIN - EFFECTS OF CURRENT-DENSITY AND CONCENTRATION ON ELECTROTRANSPORT IN-VITRO [J].
DELGADOCHARRO, MB ;
RODRIGUEZBAYON, AM ;
GUY, RH .
JOURNAL OF CONTROLLED RELEASE, 1995, 35 (01) :35-40
[7]   CHARACTERIZATION OF CONVECTIVE SOLVENT FLOW DURING IONTOPHORESIS [J].
DELGADOCHARRO, MB ;
GUY, RH .
PHARMACEUTICAL RESEARCH, 1994, 11 (07) :929-935
[8]   INVITRO AND INVIVO IONTOPHORESIS OF A TRIPEPTIDE ACROSS NUDE RAT SKIN [J].
GREEN, P ;
SHROOT, B ;
BERNERD, F ;
PILGRIM, WR ;
GUY, RH .
JOURNAL OF CONTROLLED RELEASE, 1992, 20 (03) :209-218
[9]   IONTOPHORETIC DELIVERY OF AMINO-ACIDS AND AMINO-ACID DERIVATIVES ACROSS THE SKIN INVITRO [J].
GREEN, PG ;
HINZ, RS ;
CULLANDER, C ;
YAMANE, G ;
GUY, RH .
PHARMACEUTICAL RESEARCH, 1991, 8 (09) :1113-1120
[10]   TRANSDERMAL LONTOPHORETIC PEPTIDE DELIVERY - INVITRO AND INVIVO STUDIES WITH LUTEINIZING-HORMONE-RELEASING HORMONE [J].
HEIT, MC ;
WILLIAMS, PL ;
JAYES, FL ;
CHANG, SK ;
RIVIERE, JE .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1993, 82 (03) :240-243