Synthesis of a novel heterocyclic system, imidazol[1′,2′:1,2]pyrimido[5,4-d] [1,3]thiazole

被引:4
作者
Bakavoli, M
Khodadady, A
Ghassemzadeh, M
Heravi, MM [1 ]
机构
[1] Alzahra Univ, Sch Sci, Dept Chem, Tehran, Iran
[2] Chem & Chem Engn Res Ctr Iran, Tehran, Iran
[3] Alzahra Univ, Sch Sci, Dept Chem, Tehran, Iran
关键词
imidazopyrimidothiazole; pyrimidines; carbon disulfide; tricyclic heterocycles; phrmacological importance;
D O I
10.1080/10426500108040596
中图分类号
O61 [无机化学];
学科分类号
070301 ; 081704 ;
摘要
7-Substituted amino-6-amino-2,3-dihydro-5-methylimidazo[1,2-a]pyrimidines (1) were condensed with carbon disulfide in hot pyridine to afford the novel heterocyclic system 9-methyl-1,2,6,7-tetrahydroimidazo[1',2':1,2]pyrimido[5,4-d][1,3]thiazole-2-thione (2). This compound was then converted to several substituted derivatives.
引用
收藏
页码:191 / 195
页数:5
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