The discovery and development of inhibitors of fatty acid amide hydrolase (FAAH)

被引：111

作者：

Otrubova, Katerina

Ezzili, Cyrine

Boger, Dale L. ^{[1
]}

机构：

[1] Scripps Res Inst, Dept Chem, La Jolla, CA 92037 USA

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 2011年 / 21卷 / 16期

基金：

美国国家卫生研究院;

关键词：

Fatty acid amide hydrolase; FAAH inhibitors; ALPHA-KETOHETEROCYCLE INHIBITORS; TRIFLUOROMETHYL KETONE INHIBITORS; REVERSIBLE INHIBITORS; THERAPEUTIC TARGET; MOLECULAR CHARACTERIZATION; KETOOXAZOLE INHIBITORS; EXCEPTIONALLY POTENT; BROMINE COMPOUND; IN-VITRO; ENZYME;

D O I：

10.1016/j.bmcl.2011.06.096

中图分类号：

R914 [药物化学];

学科分类号：

100705 [微生物与生化药学];

摘要：

引用

页码：4674 / 4685

页数：12

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