Conformational and spacial preferences for substrates of PepT1

被引:9
作者
Bailey, PD
Boyd, CAR
Collier, ID
George, JG
Kellett, GL
Meredith, D
Morgan, KM
Pettecrew, R
Price, RA
Pritchard, RG
机构
[1] Univ Manchester, Sch Chem, Manchester M60 1QD, Lancs, England
[2] Univ Oxford, Dept Human Anat & Genet, Oxford OX1 3QX, England
[3] Heriot Watt Univ, Dept Chem, Edinburgh EH14 4AS, Midlothian, Scotland
[4] Univ York, Dept Biol, York YO1 5DD, N Yorkshire, England
关键词
D O I
10.1039/b510697d
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
The conformation at the first residue of dipeptide substrates for the peptide transporter PepT1 has been probed using constrained peptide analogues, and the active conformation has been identified.
引用
收藏
页码:5352 / 5354
页数:3
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