A valuable heterocyclic ring transformation:: from isoxazolin-5(2H)-ones to quinolines

被引：50

作者：

Abbiati, G

Beccalli, EM

Broggini, G

Zoni, C

机构：

[1] Univ Milan, Fac Farm, Ist Chim Organ A Marchesini, I-20133 Milan, Italy

[2] Univ Insubria, Dipartimento Sci Chim Fis & Matemat, I-22100 Como, Italy

来源：

TETRAHEDRON | 2003年 / 59卷 / 50期

关键词：

quinolines; isoxazolones; catalytic hydrogenation; naphthyridine;

D O I：

10.1016/j.tet.2003.10.053

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A new synthesis of quinoline derivatives was achieved by catalytic hydrogenation of 3,4-disubstituted 2-(2-formylphenyl)isoxazolin-5(2H)-ones. In the same way, 2,3-disubstituted [1,8]naphthyridine was obtained. (C) 2003 Elsevier Ltd. All rights reserved.

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收藏

页码：9887 / 9893

页数：7

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