Synthesis and biological evaluation of cytostatin analogues

被引：27

作者：

Bialy, L

Waldmann, H

机构：

[1] Max Planck Inst Mol Physiol, Abt Chem Biol, D-44227 Dortmund, Germany

[2] Univ Dortmund, Fachbereich 3, D-44221 Dortmund, Germany

来源：

CHEMICAL COMMUNICATIONS | 2003年 / 15期

关键词：

D O I：

10.1039/b305308n

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Analogues of the serine/threonine phosphatase 2A inhibitor cytostatin were synthesized and evaluated as inhibitors of various phosphatases in order to establish a basic structure activity relationship (SAR) of the natural product.

引用

页码：1872 / 1873

页数：2

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