A convenient one-pot synthesis of 4-, 6-, and 7-azaindoles from aminopyridines

被引:18
作者
Debenham, SD [1 ]
Chan, A [1 ]
Liu, K [1 ]
Price, K [1 ]
Wood, HB [1 ]
机构
[1] Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
关键词
azaindole; aminopyridine;
D O I
10.1016/j.tetlet.2005.02.011
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
A one-pot synthesis of a variety of substituted 4-, 6-, and 7-azaindoles from commercially available aminopyridines in moderate to good yields is described. (c) 2005 Elsevier Ltd. All rights reserved.
引用
收藏
页码:2283 / 2285
页数:3
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