A3 adenosine receptors

被引:11
作者
Jacobson, KA [1 ]
Tchilibon, S [1 ]
Joshi, BV [1 ]
Gao, ZG [1 ]
机构
[1] NIDDKD, Bioorgan Chem Lab, Mol Recognit Sect, Bethesda, MD 20892 USA
来源
ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 38 | 2003年 / 38卷
关键词
D O I
10.1016/S0065-7743(03)38014-5
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:121 / 130
页数:10
相关论文
共 59 条
[1]  
Avila MY, 2002, INVEST OPHTH VIS SCI, V43, P3021
[2]   A1-, A2A- and A3-subtype adenosine receptors modulate intraocular pressure in the mouse [J].
Avila, MY ;
Stone, RA ;
Civan, MM .
BRITISH JOURNAL OF PHARMACOLOGY, 2001, 134 (02) :241-245
[3]   Resistance of muscle to tumor metastases: A role for A3 adenosine receptor agonists [J].
Bar-Yehuda, S ;
Barer, F ;
Volfsson, L ;
Fishman, P .
NEOPLASIA, 2001, 3 (02) :125-131
[4]   Synthesis, biological activity, and molecular modeling investigation of new pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as human A3 adenosine receptor antagonists [J].
Baraldi, PG ;
Cacciari, B ;
Moro, S ;
Spalluto, G ;
Pastorin, G ;
Da Ros, T ;
Klotz, KN ;
Varani, K ;
Gessi, S ;
Borea, PA .
JOURNAL OF MEDICINAL CHEMISTRY, 2002, 45 (04) :770-780
[5]   Synthesis and biological activity of a new series of N6-arylcarbamoyl, 2-(Ar)alkynyl-N6-arylcarbamoyl, and N6-carboxamido derivatives of adenosine-5′-N-ethyluronamide as A1 and A3 adenosine receptor agonists [J].
Baraldi, PG ;
Cacciari, B ;
de Las Infantas, MJP ;
Romagnoli, R ;
Spalluto, G ;
Volpini, R ;
Costanzi, S ;
Vittori, S ;
Cristalli, G ;
Melman, N ;
Park, KS ;
Ji, XD ;
Jacobson, KA .
JOURNAL OF MEDICINAL CHEMISTRY, 1998, 41 (17) :3174-3185
[6]  
BOEHRINGER INGELHEIM, 2000, Patent No. 0012511
[7]  
BOEHRINGER INGELHEIM, 2000, Patent No. 0978517
[8]  
Bowlin TL, 1997, CELL MOL BIOL, V43, P345
[9]   2-and 8-alkynyladenosines:: conformational studies and docking to human adenosine A3 receptor can explain their different biological behavior [J].
Costanzi, S ;
Lambertucci, C ;
Vittori, S ;
Volpini, R ;
Cristalli, G .
JOURNAL OF MOLECULAR GRAPHICS & MODELLING, 2003, 21 (04) :253-262
[10]   3′-aminoadenosine-5′-uronamides:: Discovery of the first highly selective agonist at the human adenosine A3 receptor [J].
DeNinno, MP ;
Masamune, H ;
Chenard, LK ;
DiRico, KJ ;
Eller, C ;
Etienne, JB ;
Tickner, JE ;
Kennedy, SP ;
Knight, DR ;
Kong, J ;
Oleynek, JJ ;
Tracey, WR ;
Hill, RJ .
JOURNAL OF MEDICINAL CHEMISTRY, 2003, 46 (03) :353-355