Synthesis of CD-ring modified 1 alpha,25-dihydroxy vitamin D analogues: E-ring analogues

被引：28

作者：

Sabbe, K

DHallewyn, C

DeClercq, P

Vandewalle, M

机构：

[1] STATE UNIV GHENT,DEPT ORGAN CHEM,ORGAN SYNTH LAB,B-9000 GHENT,BELGIUM

[2] KATHOLIEKE UNIV LEUVEN,LAB EXPTL GENEESKUNDE ENDOCRINOL,B-3030 LOUVAIN,BELGIUM

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1996年 / 6卷 / 14期

关键词：

D O I：

10.1016/0960-894X(96)00300-9

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

Vitamin D analogues, characterized by the absence of both C- and D-rings and by the presence of a five-membered ring formed by connecting C-12 and C-21 (E-ring analogues) are described. Copyright (C) 1996 Elsevier Science Ltd

引用

页码：1697 / 1702

页数：6

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