(Bromodimethyl)sulfonium bromide:: an inexpensive reagent for the solvent-free, one-pot synthesis of α-aminophosphonates

被引：70

作者：

Kudrimoti, S ^{[1
]}

Bommena, VR ^{[1
]}

机构：

[1] Indian Inst Chem Technol, Div Organ 2, Hyderabad 500007, Andhra Pradesh, India

来源：

TETRAHEDRON LETTERS | 2005年 / 46卷 / 07期

关键词：

alpha-aminophosphonates; (bromodimethyl)sulfonium; bromide; imine;

D O I：

10.1016/j.tetlet.2004.12.070

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A novel solvent-free, one-pot synthesis of alpha-aminophosphonates in the presence of catalytic (bromodimethyl)sulfonium bromide at room temperature in high yields is reported. (C) 2004 Elsevier Ltd. All rights reserved.

引用

页码：1209 / 1210

页数：2

共 28 条

[1] [Anonymous], ROLE PHOSPHONATES LI
[2] SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF ANTIBACTERIAL PHOSPHONOPEPTIDES INCORPORATING (1-AMINOETHYL)PHOSPHONIC ACID AND (AMINOMETHYL)PHOSPHONIC ACID
ATHERTON, FR
HASSALL, CH
LAMBERT, RW
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1986, 29 (01) : 29 - 40
[3] 1-AMINOALKYLPHOSPHONOUS ACIDS .1. ISOSTERES OF THE PROTEIN AMINO-ACIDS
BAYLIS, EK
CAMPBELL, CD
DINGWALL, JG
[J]. JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1984, (12): : 2845 - 2853
[4] BRUKE TR, 1994, BIOCHEM BIOPH RES CO, V204, P129
[5] BRUKE TR, 1995, J MED CHEM, V38, P1386
[6] THE SYNTHESIS OF ESTERS OF SUBSTITUTED AMINO PHOSPHONIC ACIDS
FIELDS, EK
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1952, 74 (06) : 1528 - 1531
[7] GANCARZ R, 1977, SYNTHESIS-STUTTGART, P625
[8] PHOSPHORUS AMINO-ACID-ANALOGS AS INHIBITORS OF LEUCINE AMINOPEPTIDASE
GIANNOUSIS, PP
BARTLETT, PA
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1987, 30 (09) : 1603 - 1609
[9] Kabachnik M. I., 1954, IZV AKAD NAUK K, P1024
[10] KABACHNIK MI, 1953, B ACAD SCI USSR CH+, P1126

← 1 2 3 →