Synthesis of 5-substituted 7-azaoxindoles via palladium-catalyzed reactions

被引：13

作者：

Cheung, M ^{[1
]}

Hunter, RN ^{[1
]}

Peel, MR ^{[1
]}

Lackey, KE ^{[1
]}

机构：

[1] GlaxoSmithKline, Res Triangle Pk, NC 27709 USA

来源：

HETEROCYCLES | 2001年 / 55卷 / 08期

关键词：

D O I：

10.3987/COM-01-9267

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A synthesis of 5-substituted 1,3-dihydro-2H-pyrrolo[2,3-b]pyridin-2-ones (5-substituted 7-azaoxindoles) via palladium-catalyzed Suzuki coupling, Stille coupling, and carbonylation reactions is described.

引用

页码：1583 / 1590

页数：8

共 13 条

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[4] OXIDATION OF INDOLES WITH PYRIDINIUM BROMIDE PERBROMIDE A SIMPLE AND EFFICIENT SYNTHESIS OF 7-AZAOXINDOLES
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CARTA, MP
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[8] SYNTHESIS OF 5-AZAOXINDOLE
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[9] Synthesis of substituted azaoxindoles for the preparation of aza-tenidap analogs
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