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Mechanistic considerations in high-throughput screening
被引:117
作者
:
Copeland, RA
论文数:
0
引用数:
0
h-index:
0
机构:
GlaxoSmithKline, Dept Enzymol & Mechanist Pharmacol, Collegeville, PA 19426 USA
GlaxoSmithKline, Dept Enzymol & Mechanist Pharmacol, Collegeville, PA 19426 USA
Copeland, RA
[
1
]
机构
:
[1]
GlaxoSmithKline, Dept Enzymol & Mechanist Pharmacol, Collegeville, PA 19426 USA
来源
:
ANALYTICAL BIOCHEMISTRY
|
2003年
/ 320卷
/ 01期
关键词
:
D O I
:
10.1016/S0003-2697(03)00346-4
中图分类号
:
Q5 [生物化学];
学科分类号
:
071010
[生物化学与分子生物学]
;
081704
[应用化学]
;
摘要
:
[No abstract available]
引用
收藏
页码:1 / 12
页数:12
相关论文
共 22 条
[1]
[Anonymous], TXB DRUG DESIGN DISC
[2]
Binding of nonphysiological protein and peptide substrates to proteases: Differences between urokinase-type plasminogen activator and trypsin and contributions to the evolution of regulated proteolysis
[J].
Bergstrom, RC
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, SW Med Ctr, Dept Pharmacol, Dallas, TX 75390 USA
Bergstrom, RC
;
Coombs, GS
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, SW Med Ctr, Dept Pharmacol, Dallas, TX 75390 USA
Coombs, GS
;
Ye, S
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, SW Med Ctr, Dept Pharmacol, Dallas, TX 75390 USA
Ye, S
;
Madison, EL
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, SW Med Ctr, Dept Pharmacol, Dallas, TX 75390 USA
Madison, EL
;
Goldsmith, EJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, SW Med Ctr, Dept Pharmacol, Dallas, TX 75390 USA
Goldsmith, EJ
;
Corey, DR
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, SW Med Ctr, Dept Pharmacol, Dallas, TX 75390 USA
Corey, DR
.
BIOCHEMISTRY,
2003,
42
(18)
:5395
-5402
[3]
Nematode anticoagulant protein c2 reveals a site on factor Xa that is important for macromolecular substrate binding to human prothrombinase.
[J].
Buddai, SK
论文数:
0
引用数:
0
h-index:
0
机构:
Childrens Hosp Philadelphia, Joseph Stokes Res Inst, Philadelphia, PA 19104 USA
Buddai, SK
;
Toulokhonova, L
论文数:
0
引用数:
0
h-index:
0
机构:
Childrens Hosp Philadelphia, Joseph Stokes Res Inst, Philadelphia, PA 19104 USA
Toulokhonova, L
;
Bergum, PW
论文数:
0
引用数:
0
h-index:
0
机构:
Childrens Hosp Philadelphia, Joseph Stokes Res Inst, Philadelphia, PA 19104 USA
Bergum, PW
;
Vlasuk, GP
论文数:
0
引用数:
0
h-index:
0
机构:
Childrens Hosp Philadelphia, Joseph Stokes Res Inst, Philadelphia, PA 19104 USA
Vlasuk, GP
;
Krishnaswamy, S
论文数:
0
引用数:
0
h-index:
0
机构:
Childrens Hosp Philadelphia, Joseph Stokes Res Inst, Philadelphia, PA 19104 USA
Krishnaswamy, S
.
JOURNAL OF BIOLOGICAL CHEMISTRY,
2002,
277
(29)
:26689
-26698
[4]
Copeland R. A., 2004, ENZYMES PRACTICAL IN
[5]
Is the isolated ligand binding domain a good model of the domain in the native receptor?
[J].
Deming, D
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, Hlth Sci Ctr, Dept Integrat Biol & Pharmacol, Houston, TX 77030 USA
Univ Texas, Hlth Sci Ctr, Dept Integrat Biol & Pharmacol, Houston, TX 77030 USA
Deming, D
;
Cheng, Q
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, Hlth Sci Ctr, Dept Integrat Biol & Pharmacol, Houston, TX 77030 USA
Univ Texas, Hlth Sci Ctr, Dept Integrat Biol & Pharmacol, Houston, TX 77030 USA
Cheng, Q
;
Jayaraman, V
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, Hlth Sci Ctr, Dept Integrat Biol & Pharmacol, Houston, TX 77030 USA
Univ Texas, Hlth Sci Ctr, Dept Integrat Biol & Pharmacol, Houston, TX 77030 USA
Jayaraman, V
.
JOURNAL OF BIOLOGICAL CHEMISTRY,
2003,
278
(20)
:17589
-17592
[6]
Drug discovery: A historical perspective
[J].
Drews, J
论文数:
0
引用数:
0
h-index:
0
机构:
Int Biomed Management Partners, Basel, Switzerland
Int Biomed Management Partners, Basel, Switzerland
Drews, J
.
SCIENCE,
2000,
287
(5460)
:1960
-1964
[7]
Identification of a novel inhibitor of mitogen-activated protein kinase kinase
[J].
Favata, MF
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Favata, MF
;
Horiuchi, KY
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Horiuchi, KY
;
Manos, EJ
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Manos, EJ
;
Daulerio, AJ
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Daulerio, AJ
;
Stradley, DA
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Stradley, DA
;
Feeser, WS
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Feeser, WS
;
Van Dyk, DE
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Van Dyk, DE
;
Pitts, WJ
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Pitts, WJ
;
Earl, RA
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Earl, RA
;
Hobbs, F
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Hobbs, F
;
Copeland, RA
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Copeland, RA
;
Magolda, RL
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Magolda, RL
;
Scherle, PA
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Scherle, PA
;
Trzaskos, JM
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Trzaskos, JM
.
JOURNAL OF BIOLOGICAL CHEMISTRY,
1998,
273
(29)
:18623
-18632
[8]
Mutagenesis and mechanism-based inhibition of Streptococcus pyogenes Glu-tRNAGln amidotransferase implicate a serine-based glutaminase site
[J].
Harpel, MR
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Harpel, MR
;
Horiuchi, KIY
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Horiuchi, KIY
;
Luo, Y
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Luo, Y
;
Shen, L
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Shen, L
;
Jiang, WJ
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Jiang, WJ
;
Nelson, DJ
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Nelson, DJ
;
Kelley, CRC
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Kelley, CRC
;
Decicco, CP
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Decicco, CP
;
Copeland, RA
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Copeland, RA
.
BIOCHEMISTRY,
2002,
41
(20)
:6398
-6407
[9]
DOES ANY ENZYME FOLLOW MICHAELIS-MENTEN EQUATION
[J].
HILL, CM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV MANCHESTER,ST MARYS HOSP,DEPT OBSTET & GYNAECOL,MANCHESTER M13 0JH,ENGLAND
UNIV MANCHESTER,ST MARYS HOSP,DEPT OBSTET & GYNAECOL,MANCHESTER M13 0JH,ENGLAND
HILL, CM
;
WAIGHT, RD
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV MANCHESTER,ST MARYS HOSP,DEPT OBSTET & GYNAECOL,MANCHESTER M13 0JH,ENGLAND
UNIV MANCHESTER,ST MARYS HOSP,DEPT OBSTET & GYNAECOL,MANCHESTER M13 0JH,ENGLAND
WAIGHT, RD
;
论文数:
引用数:
h-index:
机构:
BARDSLEY, WG
.
MOLECULAR AND CELLULAR BIOCHEMISTRY,
1977,
15
(03)
:173
-178
[10]
Competitive inhibition of MAP kinase activation by a peptide representing the αc helix of ERK
[J].
Horiuchi, KY
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Pharmaceut Co, Res Labs, Chem Enzymol, Wilmington, DE 19880 USA
Horiuchi, KY
;
Scherle, PA
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Pharmaceut Co, Res Labs, Chem Enzymol, Wilmington, DE 19880 USA
Scherle, PA
;
Trzaskos, JM
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Pharmaceut Co, Res Labs, Chem Enzymol, Wilmington, DE 19880 USA
Trzaskos, JM
;
Copeland, RA
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Pharmaceut Co, Res Labs, Chem Enzymol, Wilmington, DE 19880 USA
Copeland, RA
.
BIOCHEMISTRY,
1998,
37
(25)
:8879
-8885
←
1
2
3
→
共 22 条
[1]
[Anonymous], TXB DRUG DESIGN DISC
[2]
Binding of nonphysiological protein and peptide substrates to proteases: Differences between urokinase-type plasminogen activator and trypsin and contributions to the evolution of regulated proteolysis
[J].
Bergstrom, RC
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, SW Med Ctr, Dept Pharmacol, Dallas, TX 75390 USA
Bergstrom, RC
;
Coombs, GS
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, SW Med Ctr, Dept Pharmacol, Dallas, TX 75390 USA
Coombs, GS
;
Ye, S
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, SW Med Ctr, Dept Pharmacol, Dallas, TX 75390 USA
Ye, S
;
Madison, EL
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, SW Med Ctr, Dept Pharmacol, Dallas, TX 75390 USA
Madison, EL
;
Goldsmith, EJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, SW Med Ctr, Dept Pharmacol, Dallas, TX 75390 USA
Goldsmith, EJ
;
Corey, DR
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, SW Med Ctr, Dept Pharmacol, Dallas, TX 75390 USA
Corey, DR
.
BIOCHEMISTRY,
2003,
42
(18)
:5395
-5402
[3]
Nematode anticoagulant protein c2 reveals a site on factor Xa that is important for macromolecular substrate binding to human prothrombinase.
[J].
Buddai, SK
论文数:
0
引用数:
0
h-index:
0
机构:
Childrens Hosp Philadelphia, Joseph Stokes Res Inst, Philadelphia, PA 19104 USA
Buddai, SK
;
Toulokhonova, L
论文数:
0
引用数:
0
h-index:
0
机构:
Childrens Hosp Philadelphia, Joseph Stokes Res Inst, Philadelphia, PA 19104 USA
Toulokhonova, L
;
Bergum, PW
论文数:
0
引用数:
0
h-index:
0
机构:
Childrens Hosp Philadelphia, Joseph Stokes Res Inst, Philadelphia, PA 19104 USA
Bergum, PW
;
Vlasuk, GP
论文数:
0
引用数:
0
h-index:
0
机构:
Childrens Hosp Philadelphia, Joseph Stokes Res Inst, Philadelphia, PA 19104 USA
Vlasuk, GP
;
Krishnaswamy, S
论文数:
0
引用数:
0
h-index:
0
机构:
Childrens Hosp Philadelphia, Joseph Stokes Res Inst, Philadelphia, PA 19104 USA
Krishnaswamy, S
.
JOURNAL OF BIOLOGICAL CHEMISTRY,
2002,
277
(29)
:26689
-26698
[4]
Copeland R. A., 2004, ENZYMES PRACTICAL IN
[5]
Is the isolated ligand binding domain a good model of the domain in the native receptor?
[J].
Deming, D
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, Hlth Sci Ctr, Dept Integrat Biol & Pharmacol, Houston, TX 77030 USA
Univ Texas, Hlth Sci Ctr, Dept Integrat Biol & Pharmacol, Houston, TX 77030 USA
Deming, D
;
Cheng, Q
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, Hlth Sci Ctr, Dept Integrat Biol & Pharmacol, Houston, TX 77030 USA
Univ Texas, Hlth Sci Ctr, Dept Integrat Biol & Pharmacol, Houston, TX 77030 USA
Cheng, Q
;
Jayaraman, V
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas, Hlth Sci Ctr, Dept Integrat Biol & Pharmacol, Houston, TX 77030 USA
Univ Texas, Hlth Sci Ctr, Dept Integrat Biol & Pharmacol, Houston, TX 77030 USA
Jayaraman, V
.
JOURNAL OF BIOLOGICAL CHEMISTRY,
2003,
278
(20)
:17589
-17592
[6]
Drug discovery: A historical perspective
[J].
Drews, J
论文数:
0
引用数:
0
h-index:
0
机构:
Int Biomed Management Partners, Basel, Switzerland
Int Biomed Management Partners, Basel, Switzerland
Drews, J
.
SCIENCE,
2000,
287
(5460)
:1960
-1964
[7]
Identification of a novel inhibitor of mitogen-activated protein kinase kinase
[J].
Favata, MF
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Favata, MF
;
Horiuchi, KY
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Horiuchi, KY
;
Manos, EJ
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Manos, EJ
;
Daulerio, AJ
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Daulerio, AJ
;
Stradley, DA
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Stradley, DA
;
Feeser, WS
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Feeser, WS
;
Van Dyk, DE
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Van Dyk, DE
;
Pitts, WJ
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Pitts, WJ
;
Earl, RA
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Earl, RA
;
Hobbs, F
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Hobbs, F
;
Copeland, RA
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Copeland, RA
;
Magolda, RL
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Magolda, RL
;
Scherle, PA
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Scherle, PA
;
Trzaskos, JM
论文数:
0
引用数:
0
h-index:
0
机构:
Dupont Merck Res Labs, Inflammatory Dis Res, Wilmington, DE 19880 USA
Trzaskos, JM
.
JOURNAL OF BIOLOGICAL CHEMISTRY,
1998,
273
(29)
:18623
-18632
[8]
Mutagenesis and mechanism-based inhibition of Streptococcus pyogenes Glu-tRNAGln amidotransferase implicate a serine-based glutaminase site
[J].
Harpel, MR
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Harpel, MR
;
Horiuchi, KIY
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Horiuchi, KIY
;
Luo, Y
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Luo, Y
;
Shen, L
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Shen, L
;
Jiang, WJ
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Jiang, WJ
;
Nelson, DJ
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Nelson, DJ
;
Kelley, CRC
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Kelley, CRC
;
Decicco, CP
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Decicco, CP
;
Copeland, RA
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Co, Expt Stn, Dept Chem Enzymol, Wilmington, DE 19880 USA
Copeland, RA
.
BIOCHEMISTRY,
2002,
41
(20)
:6398
-6407
[9]
DOES ANY ENZYME FOLLOW MICHAELIS-MENTEN EQUATION
[J].
HILL, CM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV MANCHESTER,ST MARYS HOSP,DEPT OBSTET & GYNAECOL,MANCHESTER M13 0JH,ENGLAND
UNIV MANCHESTER,ST MARYS HOSP,DEPT OBSTET & GYNAECOL,MANCHESTER M13 0JH,ENGLAND
HILL, CM
;
WAIGHT, RD
论文数:
0
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