Efficient syntheses of 4-iodopyridine and of 4-pyridylboronic acid pinacol ester

被引：70

作者：

Coudret, C

机构：

[1] Molecular Electronics Group, CEMES, CNRS, 31055 Toulouse Cedex

来源：

SYNTHETIC COMMUNICATIONS | 1996年 / 26卷 / 19期

关键词：

D O I：

10.1080/00397919608003763

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

4-iodopyridine can be prepared in good yield by low temperature diazotation-Sandmeyer reaction of the corresponding amine, then efficiently converted to the air-stable pinacol ester of 4-pyridylboronic acid.

引用

页码：3543 / 3547

页数：5

共 15 条

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