A new and convenient synthesis of some substituted thiohydantoins

被引:11
作者
Dürüst, Y [1 ]
Nohut, F [1 ]
机构
[1] Kocaeli Univ, Fac Arts & Sci, Dept Chem, TR-41300 Izmit, Turkey
关键词
D O I
10.1080/00397919908086188
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
3-Substituted thiohydantoins (2a-g) were synthesized in satisfactory yields by the reaction of N-substituted thioureas (1a-g) with chloroacetylchloride in the presence of triethylamine under reflux in dioxane. S-Alkylated products (7, 8) were! obtained from the reaction of 3-p-tolyl -thiohydantoin (2d) with p-nitrobenzylchloride and 3-phenyl-5-chloromethyl-1,2,4-oxadiazole.
引用
收藏
页码:1997 / 2005
页数:9
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