Rapid synthesis of α-ketoamides using microwave irradiation-simultaneous cooling method

被引：97

作者：

Chen, JJ ^{[1
]}

Deshpande, SV ^{[1
]}

机构：

[1] Procter & Gamble Pharmaceut, Mason, OH 45040 USA

来源：

关键词：

microwave synthesis; alpha-ketoamide; isocyanide chemistry;

D O I：

10.1016/j.tetlet.2003.09.180

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：8873 / 8876

页数：4

共 27 条

[1] BECK Y, 1989, TRANSPLANT P, V21, P3464
[2] FK506 AND RAPAMYCIN - NOVEL PHARMACOLOGICAL PROBES OF THE IMMUNE-RESPONSE
CHANG, JY
SEHGAL, SN
BANSBACH, CC
[J]. TRENDS IN PHARMACOLOGICAL SCIENCES, 1991, 12 (06) : 218 - 223
[3] Ganesh V, 1996, PROTEIN SCI, V5, P825
[4] Glycine α-ketoamides as HCVNS3 protease inhibitors
Han, W
Hu, ZL
Jiang, XJ
Wasserman, ZR
Decicco, CP
[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2003, 13 (06) : 1111 - 1114
[5] Hayes B.L., 2002, MICROWAVE SYNTHESIS
[6] KAY JE, 1991, IMMUNOLOGY, V72, P544
[7] Potent and selective nonpeptide inhibitors of caspases 3 and 7
Lee, D
Long, SA
Murray, JH
Adams, JL
Nuttall, ME
Nadeau, DP
Kikly, K
Winkler, JD
Sung, CM
Ryan, MD
Levy, MA
Keller, PM
DeWolf, WE
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 2001, 44 (12) : 2015 - 2026
[8] INHIBITION OF THROMBIN AND OTHER TRYPSIN-LIKE SERINE PROTEINASES BY CYCLOTHEONAMIDE-A
LEWIS, SD
NG, AS
BALDWIN, JJ
FUSETANI, N
NAYLOR, AM
SHAFER, JA
[J]. THROMBOSIS RESEARCH, 1993, 70 (02) : 173 - 190
[9] PEPTIDE ALPHA-KETO ESTER, ALPHA-KETO AMIDE, AND ALPHA-KETO ACID INHIBITORS OF CALPAINS AND OTHER CYSTEINE PROTEASES
LI, ZZ
PATIL, GS
GOLUBSKI, ZE
HORI, H
TEHRANI, K
FOREMAN, JE
EVELETH, DD
BARTUS, RT
POWERS, JC
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1993, 36 (22) : 3472 - 3480
[10] Microwave assisted organic synthesis -: a review
Lidström, P
Tierney, J
Wathey, B
Westman, J
[J]. TETRAHEDRON, 2001, 57 (45) : 9225 - 9283