A facile total synthesis of rutaecarpine

被引：42

作者：

Chavan, SP ^{[1
]}

Sivappa, R ^{[1
]}

机构：

[1] Natl Chem Lab, Div Organ Chem Technol, Pune 411008, Maharashtra, India

来源：

TETRAHEDRON LETTERS | 2004年 / 45卷 / 05期

关键词：

rutaecarpine; indoloquinazoline alkaloid; Dieckmann condensation-decarboxylation;

D O I：

10.1016/j.tetlet.2003.11.090

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The indoloquinazoline alkaloid rutaecarpine has been synthesized efficiently by employing 9,10,11,12-tetrahydro-4H-pyrido[2,1-b]quinazoline-4,9-dione (4) as a key intermediate, which was prepared by adapting a Dieckmann condensation-decarboxylation sequence from quinazolinone diester 6. (C) 2003 Elsevier Ltd. All rights reserved.

引用

页码：997 / 999

页数：3

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