Synthesis of a photoactivatable probe of the anandamide re-uptake

被引：4

作者：

Balas, L ^{[1
]}

Hellal, M ^{[1
]}

Rossi, JC ^{[1
]}

Durand, T ^{[1
]}

机构：

[1] Fac Pharm Montpellier, CNRS, UMR 5074, F-34093 Montpellier, France

来源：

NATURAL PRODUCT RESEARCH | 2005年 / 19卷 / 04期

关键词：

anandamide re-uptake; iodo-arylazido probe; endocannabinoid system;

D O I：

10.1080/14786410500057015

中图分类号：

O69 [应用化学];

学科分类号：

081704 ;

摘要：

To date, despite extensive investigations, full understanding of the endocannabinoid system remains elusive; in particular, anandamide cellular uptake is a current controversial topic. An iodo-arylazido probe was synthesized from commercially available azelaic acid monomethyl ester, in order to shed light on the anandamide transport process.

引用

页码：419 / 423

页数：5

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