Isochroman-6-carboxamides as highly selective 5-HT1D agonists:: Potential new treatment for migraine without cardiovascular side effects

被引:81
作者
Ennis, MD [1 ]
Ghazal, NB
Hoffman, RL
Smith, MW
Schlachter, SK
Lawson, CF
Bin Im, W
Pregenzer, JF
Svensson, KA
Lewis, RA
Hall, ED
Sutter, DM
Harris, LT
McCall, RB
机构
[1] Pharmacia & Upjohn Inc, Struct Analyt & Med Chem, Kalamazoo, MI 49001 USA
[2] Pharmacia & Upjohn Inc, Discovery Technol, Kalamazoo, MI 49001 USA
[3] Pharmacia & Upjohn Inc, CNS Dis Res, Kalamazoo, MI 49001 USA
[4] Pharmacia & Upjohn Inc, Cardiovasc Pharmacol, Kalamazoo, MI 49001 USA
关键词
D O I
10.1021/jm980137o
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:2180 / 2183
页数:4
相关论文
共 19 条