Second joint French-Swiss meeting on medicinal chemistry

被引:2
作者
Froestl, W [1 ]
机构
[1] Novartis Pharma AG, CH-4002 Basel, Switzerland
关键词
conference report; french-swiss meeting; g-protein coupled receptors; protein kinase inhibitors; oncology research;
D O I
10.2533/000942904777678280
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
引用
收藏
页码:54 / 61
页数:8
相关论文
共 39 条
[1]  
Altmann KH, 2002, HELV CHIM ACTA, V85, P4086, DOI 10.1002/1522-2675(200211)85:11<4086::AID-HLCA4086>3.0.CO
[2]  
2-7
[3]   New selective ligands of human cloned melatonin MT1 and MT2 receptors [J].
Audinot, V ;
Mailliet, F ;
Lahaye-Brasseur, C ;
Bonnaud, A ;
Le Gall, A ;
Amossé, C ;
Dromaint, S ;
Rodriguez, M ;
Nagel, N ;
Galizzi, JP ;
Malpaux, B ;
Guillaumet, G ;
Lesieur, D ;
Lefoulon, F ;
Renard, P ;
Delagrange, P ;
Boutin, JA .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 2003, 367 (06) :553-561
[4]   Protein-based virtual screening of chemical databases. II. Are homology models of G-protein coupled receptors suitable targets? [J].
Bissantz, C ;
Bernard, P ;
Hibert, M ;
Rognan, D .
PROTEINS-STRUCTURE FUNCTION AND BIOINFORMATICS, 2003, 50 (01) :5-25
[5]   Traceless solid-phase synthesis of 2,6,9-trisubstituted purines from resin bound 6-thiopurines [J].
Brun, V ;
Legraverend, M ;
Grierson, DS .
TETRAHEDRON, 2002, 58 (39) :7911-7923
[6]  
Brun V, 2001, TETRAHEDRON LETT, V42, P8169, DOI 10.1016/S0040-4039(01)01753-1
[7]   Cyclin-dependent kinase (CDK) inhibitors: development of a general strategy for the construction of 2,6,9-trisubstituted purine libraries. Part I [J].
Brun, V ;
Legraverend, M ;
Grierson, DS .
TETRAHEDRON LETTERS, 2001, 42 (46) :8161-8164
[8]  
Brun V, 2001, TETRAHEDRON LETT, V42, P8165, DOI 10.1016/S0040-4039(01)01752-X
[9]   Glivec (ST1571, Imatinib), a rationally developed, targeted anticancer drug [J].
Capdeville, R ;
Buchdunger, E ;
Zimmermann, J ;
Matter, A .
NATURE REVIEWS DRUG DISCOVERY, 2002, 1 (07) :493-502
[10]   Structure-based screening of low-affinity compounds [J].
Carr, R ;
Jhoti, H .
DRUG DISCOVERY TODAY, 2002, 7 (09) :522-527