Labelled sigma receptor ligands: can their role in neurology and oncology be extended?

被引:25
作者
Caveliers, V
Everaert, H
Lahoutte, T
Dierickx, LO
John, CS
Bossuyt, A
机构
[1] Free Univ Hosp Brussels, AZ, Dept Nucl Med, B-1090 Brussels, Belgium
[2] George Washington Univ, Dept Radiol, Washington, DC 20052 USA
关键词
D O I
10.1007/s002590000368
中图分类号
R8 [特种医学]; R445 [影像诊断学];
学科分类号
1002 ; 100207 ; 1009 ;
摘要
引用
收藏
页码:133 / 135
页数:3
相关论文
共 28 条
[1]   Effect of ploidy, recruitment, environmental factors, and tamoxifen treatment on the expression of sigma-2 receptors in proliferating and quiescent tumour cells [J].
Al-Nabulsi, I ;
Mach, RH ;
Wang, LM ;
Wallen, CA ;
Keng, PC ;
Sten, K ;
Childers, SR ;
Wheeler, KT .
BRITISH JOURNAL OF CANCER, 1999, 81 (06) :925-933
[2]  
BEM WT, 1991, CANCER RES, V51, P6558
[3]  
Bowen W D, 2000, Pharm Acta Helv, V74, P211
[4]   EVIDENCE FOR A MULTI-SITE MODEL OF THE RAT-BRAIN SIGMA-RECEPTOR [J].
BOWEN, WD ;
HELLEWELL, SB ;
MCGARRY, KA .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1989, 163 (2-3) :309-318
[5]  
Everaert H, 1997, J NUCL MED, V38, P870
[6]  
Everaert H, 1997, ANTICANCER RES, V17, P1577
[7]   SIGMA-RECEPTORS - FROM MOLECULE TO MAN [J].
FERRIS, CD ;
HIRSCH, DJ ;
BROOKS, BP ;
SNYDER, SH .
JOURNAL OF NEUROCHEMISTRY, 1991, 57 (03) :729-737
[8]   Purification, molecular cloning, and expression of the mammalian sigma(1)-binding site [J].
Hanner, M ;
Moebius, FF ;
Flandorfer, A ;
Knaus, HG ;
Striessnig, J ;
Kempner, E ;
Glossmann, H .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1996, 93 (15) :8072-8077
[9]   A SIGMA-LIKE BINDING-SITE IN RAT PHEOCHROMOCYTOMA (PC12) CELLS - DECREASED AFFINITY FOR (+)-BENZOMORPHANS AND LOWER MOLECULAR-WEIGHT SUGGEST A DIFFERENT SIGMA RECEPTOR FORM FROM THAT OF GUINEA-PIG BRAIN [J].
HELLEWELL, SB ;
BOWEN, WD .
BRAIN RESEARCH, 1990, 527 (02) :244-253
[10]   RAT-LIVER AND KIDNEY CONTAIN HIGH-DENSITIES OF SIGMA(1) AND SIGMA(2) RECEPTORS - CHARACTERIZATION BY LIGAND-BINDING AND PHOTOAFFINITY-LABELING [J].
HELLEWELL, SB ;
BRUCE, A ;
FEINSTEIN, G ;
ORRINGER, J ;
WILLIAMS, W ;
BOWEN, WD .
EUROPEAN JOURNAL OF PHARMACOLOGY-MOLECULAR PHARMACOLOGY SECTION, 1994, 268 (01) :9-18