Syntheses of carboranylpyrroles

被引：18

作者：

Chayer, S

Jaquinod, L

Smith, KM

Vicente, MGH

机构：

[1] Univ Calif Davis, Dept Chem, Davis, CA 95616 USA

[2] Univ Calif Davis, Dept Neurol Surg, Davis, CA 95616 USA

来源：

TETRAHEDRON LETTERS | 2001年 / 42卷 / 44期

基金：

美国国家卫生研究院;

关键词：

D O I：

10.1016/S0040-4039(01)01675-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The syntheses of three carboranylpyrroles (5, 10 and 14) bearing carborane cages in 3-position and/or 4-position of the pyrrole ring, either directly linked or through a methylene spacer, are described. Tetramerization of two carboranylpyrroles afforded the corresponding beta -carboranylporphyrins, as mixtures of type I IV isomers. (C) 2001 Elsevier Science Ltd. All rights reserved.

引用

收藏

页码：7759 / 7761

页数：3

相关论文

共 21 条

[1] 3-CHLORO-2-(PHENYLSULFINYL)-1-PROPENE AND 3-CHLORO-2-(PHENYLSULFONYL)-1-PROPENE - PREPARATION AND UTILITY AS REAGENTS FOR ALPHA,ALPHA'-ANNELATION OF CYCLIC-KETONES [J].

ANZEVENO, PB ;

MATTHEWS, DP ;

BARNEY, CL ;

BARBUCH, RJ .

JOURNAL OF ORGANIC CHEMISTRY, 1984, 49 (17) :3134-3138

[2] THE PREPARATION OF PYRROLE-2-CARBOXYLATES FROM VINYL SULFONES [J].

ARNOLD, DP ;

BURGESSDEAN, L ;

HUBBARD, J ;

RAHMAN, MA .

AUSTRALIAN JOURNAL OF CHEMISTRY, 1994, 47 (05) :969-974

[3] Boron neutron capture therapy of brain tumors: An emerging therapeutic modality [J].

Barth, RF ;

Soloway, AH ;

Goodman, JH ;

Gahbauer, RA ;

Gupta, N ;

Blue, TE ;

Yang, WL ;

Tjarks, W .

NEUROSURGERY, 1999, 44 (03) :433-450

[4]

BARTON DHR, 1990, TETRAHEDRON, V46, P7587

[5] A USEFUL PREPARATION OF PYRROLES FROM ALPHA,BETA-UNSATURATED SULFONES [J].

HAAKE, G ;

STRUVE, D ;

MONTFORTS, FP .

TETRAHEDRON LETTERS, 1994, 35 (52) :9703-9704

[6] STUDIES ON THE ANTITUMOR AGENT-CC-1065 1-PHENYLSULFONYL-1,3-BUTADIENE - AN ELECTROPHILIC EQUIVALENT TO 1,3-BUTADIENE FOR THE SYNTHESIS OF 3,31-BIPYRROLES [J].

HALAZY, S ;

MAGNUS, P .

TETRAHEDRON LETTERS, 1984, 25 (14) :1421-1424

[7] SELECTIVE TUMOR UPTAKE OF A BORONATED PORPHYRIN IN AN ANIMAL-MODEL OF CEREBRAL GLIOMA [J].

HILL, JS ;

KAHL, SB ;

KAYE, AH ;

STYLLI, SS ;

KOO, MS ;

GONZALES, MF ;

VARDAXIS, NJ ;

JOHNSON, CI .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1992, 89 (05) :1785-1789

[8] Effect of dose and infusion time on the delivery of p-boronophenylalanine for neutron capture therapy [J].

Joel, DD ;

Coderre, JA ;

Micca, PL ;

Nawrocky, MM .

JOURNAL OF NEURO-ONCOLOGY, 1999, 41 (03) :213-221

[9] LITHIUM IODIDE-CATALYZED ALKYLATION OF CARBORANES [J].

KABALKA, GW ;

REDDY, NK ;

NARAYANA, C .

TETRAHEDRON LETTERS, 1992, 33 (50) :7687-7688

[10] Pharmacokinetics and boron uptake of BSH (Na2B12H11SH) in patients with intracranial tumors [J].

Kageji, T ;

Nakagawa, Y ;

Kitamura, K ;

Matsumoto, K ;

Hatanaka, H .

JOURNAL OF NEURO-ONCOLOGY, 1997, 33 (1-2) :117-130