ν-triazolines.: Part 41.: A new synthesis of 2-alkylquinazolines and 2,9-dialkylpyrimido[4,5-b]indoles

被引：17

作者：

Erba, E

Pocar, D

Valle, M

机构：

[1] Univ Milan, Fac Farm, Ist Chim Organ, I-20133 Milan, Italy

[2] Univ Milan, Ctr Interuniv Ric Reaz Pericicliche & Sintesi Sis, I-20133 Milan, Italy

来源：

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 1999年 / 04期

关键词：

D O I：

10.1039/a809321k

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

2-Alkylquinazolines were obtained from amidines by reaction with ammonia. The synthesis has been applied to the preparation of 2,9-dialkylpyrimido[4,5-b]indoles, in a one pot reaction, from 1-alkyl-2-azidoindole-3-carbaldehydes, a secondary amine and aldehydes and reaction with ammonia.

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页码：421 / 425

页数：5

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