This review centers on recent findings with respect to modulating cancer multidrug resistance (MDR) with the well-known flavonoid quercetin. After a short introduction of quercetin, major in vitro and in vivo findings are summarized showing that quercetin is a MDR modulator and thus a potential chemosensitizer. Finally, we contemplate future prospects of modulating MDR in the clinic. (C) 2010 Elsevier Inc. All rights reserved.
机构:
Unilever Res Labs, Unilever Hlth Inst, NL-3130 AC Vlaardingen, NetherlandsUnilever Res Labs, Unilever Hlth Inst, NL-3130 AC Vlaardingen, Netherlands
Abrahamse, SL
;
Kloots, WJ
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Unilever Res Labs, Unilever Hlth Inst, NL-3130 AC Vlaardingen, NetherlandsUnilever Res Labs, Unilever Hlth Inst, NL-3130 AC Vlaardingen, Netherlands
Kloots, WJ
;
van Amelsvoort, JMM
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Unilever Res Labs, Unilever Hlth Inst, NL-3130 AC Vlaardingen, NetherlandsUnilever Res Labs, Unilever Hlth Inst, NL-3130 AC Vlaardingen, Netherlands
机构:
Dabur Res Fdn, Ghaziabad 201010, UP, India
Hamdard Univ, Dept Pharmaceut, Fac Pharm, New Delhi 110062, IndiaDabur Res Fdn, Ghaziabad 201010, UP, India
Bansal, Tripta
;
Awasthi, Anshumali
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Dabur Res Fdn, Ghaziabad 201010, UP, IndiaDabur Res Fdn, Ghaziabad 201010, UP, India
Awasthi, Anshumali
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Jaggi, Manu
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Dabur Res Fdn, Ghaziabad 201010, UP, IndiaDabur Res Fdn, Ghaziabad 201010, UP, India
Jaggi, Manu
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Khar, Roop K.
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Hamdard Univ, Dept Pharmaceut, Fac Pharm, New Delhi 110062, IndiaDabur Res Fdn, Ghaziabad 201010, UP, India
Khar, Roop K.
;
Talegaonkar, Sushama
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Hamdard Univ, Dept Pharmaceut, Fac Pharm, New Delhi 110062, IndiaDabur Res Fdn, Ghaziabad 201010, UP, India
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Unilever Res Labs, Unilever Hlth Inst, NL-3130 AC Vlaardingen, NetherlandsUnilever Res Labs, Unilever Hlth Inst, NL-3130 AC Vlaardingen, Netherlands
Abrahamse, SL
;
Kloots, WJ
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Unilever Res Labs, Unilever Hlth Inst, NL-3130 AC Vlaardingen, NetherlandsUnilever Res Labs, Unilever Hlth Inst, NL-3130 AC Vlaardingen, Netherlands
Kloots, WJ
;
van Amelsvoort, JMM
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Unilever Res Labs, Unilever Hlth Inst, NL-3130 AC Vlaardingen, NetherlandsUnilever Res Labs, Unilever Hlth Inst, NL-3130 AC Vlaardingen, Netherlands
机构:
Dabur Res Fdn, Ghaziabad 201010, UP, India
Hamdard Univ, Dept Pharmaceut, Fac Pharm, New Delhi 110062, IndiaDabur Res Fdn, Ghaziabad 201010, UP, India
Bansal, Tripta
;
Awasthi, Anshumali
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Dabur Res Fdn, Ghaziabad 201010, UP, IndiaDabur Res Fdn, Ghaziabad 201010, UP, India
Awasthi, Anshumali
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Jaggi, Manu
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Dabur Res Fdn, Ghaziabad 201010, UP, IndiaDabur Res Fdn, Ghaziabad 201010, UP, India
Jaggi, Manu
;
Khar, Roop K.
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机构:
Hamdard Univ, Dept Pharmaceut, Fac Pharm, New Delhi 110062, IndiaDabur Res Fdn, Ghaziabad 201010, UP, India
Khar, Roop K.
;
Talegaonkar, Sushama
论文数: 0引用数: 0
h-index: 0
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Hamdard Univ, Dept Pharmaceut, Fac Pharm, New Delhi 110062, IndiaDabur Res Fdn, Ghaziabad 201010, UP, India