Data base of three-dimensional structures of HIV proteinases

被引:43
作者
Vondrasek, J [1 ]
vanBuskirk, CP [1 ]
Wlodawer, A [1 ]
机构
[1] JOHNS HOPKINS UNIV,KRIEGER MIND BRAIN INST,BALTIMORE,MD 21218
关键词
D O I
10.1038/nsb0197-8
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:8 / 8
页数:1
相关论文
共 10 条
  • [1] ABT-538 IS A POTENT INHIBITOR OF HUMAN-IMMUNODEFICIENCY-VIRUS PROTEASE AND HAS HIGH ORAL BIOAVAILABILITY IN HUMANS
    KEMPF, DJ
    MARSH, KC
    DENISSEN, JF
    MCDONALD, E
    VASAVANONDA, S
    FLENTGE, CA
    GREEN, BE
    FINO, L
    PARK, CH
    KONG, XP
    WIDEBURG, NE
    SALDIVAR, A
    RUIZ, L
    KATI, WM
    SHAM, HL
    ROBINS, T
    STEWART, KD
    HSU, A
    PLATTNER, JJ
    LEONARD, JM
    NORBECK, DW
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1995, 92 (07) : 2484 - 2488
  • [2] MARTIN ACR, 1996, PROFIT
  • [3] 3-DIMENSIONAL STRUCTURE OF ASPARTYL PROTEASE FROM HUMAN IMMUNODEFICIENCY VIRUS HIV-1
    NAVIA, MA
    FITZGERALD, PMD
    MCKEEVER, BM
    LEU, CT
    HEIMBACH, JC
    HERBER, WK
    SIGAL, IS
    DARKE, PL
    SPRINGER, JP
    [J]. NATURE, 1989, 337 (6208) : 615 - 620
  • [4] PROTEIN STRUCTURE-BASED DESIGN OF POTENT ORALLY BIOAVAILABLE, NONPEPTIDE INHIBITORS OF HUMAN-IMMUNODEFICIENCY-VIRUS PROTEASE
    REICH, SH
    MELNICK, M
    DAVIES, JF
    APPELT, K
    LEWIS, KK
    FUHRY, MA
    PINO, M
    TRIPPE, AJ
    NGUYEN, D
    DAWSON, H
    WU, BW
    MUSICK, L
    KOSA, M
    KAHIL, D
    WEBBER, S
    GEHLHAAR, DK
    ANDRADA, D
    SHETTY, B
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1995, 92 (08) : 3298 - 3302
  • [5] RASMOL - BIOMOLECULAR GRAPHICS FOR ALL
    SAYLE, RA
    MILNERWHITE, EJ
    [J]. TRENDS IN BIOCHEMICAL SCIENCES, 1995, 20 (09) : 374 - 376
  • [6] SHOICHET BK, 1993, PROTEIN ENG, V6, P223
  • [7] Vondrasek J, 1996, SCIENCE, V272, P337
  • [8] Winslow D L, 1995, AIDS, V9 Suppl A, pS183
  • [9] STRUCTURE-BASED INHIBITORS OF HIV-1 PROTEASE
    WLODAWER, A
    ERICKSON, JW
    [J]. ANNUAL REVIEW OF BIOCHEMISTRY, 1993, 62 : 543 - 585
  • [10] CONSERVED FOLDING IN RETROVIRAL PROTEASES - CRYSTAL-STRUCTURE OF A SYNTHETIC HIV-1 PROTEASE
    WLODAWER, A
    MILLER, M
    JASKOLSKI, M
    SATHYANARAYANA, BK
    BALDWIN, E
    WEBER, IT
    SELK, LM
    CLAWSON, L
    SCHNEIDER, J
    KENT, SBH
    [J]. SCIENCE, 1989, 245 (4918) : 616 - 621