共 8 条
[1]
A small molecule-kinase interaction map for clinical kinase inhibitors
[J].
Fabian, MA
;
Biggs, WH
;
Treiber, DK
;
Atteridge, CE
;
Azimioara, MD
;
Benedetti, MG
;
Carter, TA
;
Ciceri, P
;
Edeen, PT
;
Floyd, M
;
Ford, JM
;
Galvin, M
;
Gerlach, JL
;
Grotzfeld, RM
;
Herrgard, S
;
Insko, DE
;
Insko, MA
;
Lai, AG
;
Lélias, JM
;
Mehta, SA
;
Milanov, ZV
;
Velasco, AM
;
Wodicka, LM
;
Patel, HK
;
Zarrinkar, PP
;
Lockhart, DJ
.
NATURE BIOTECHNOLOGY,
2005, 23 (03)
:329-336

Fabian, MA
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Biggs, WH
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Treiber, DK
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Atteridge, CE
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Azimioara, MD
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Benedetti, MG
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Carter, TA
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Ciceri, P
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Edeen, PT
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Floyd, M
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Ford, JM
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Galvin, M
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Gerlach, JL
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Grotzfeld, RM
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Herrgard, S
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Insko, DE
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Insko, MA
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Lai, AG
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Lélias, JM
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Mehta, SA
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Milanov, ZV
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Velasco, AM
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Wodicka, LM
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Patel, HK
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Zarrinkar, PP
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA

Lockhart, DJ
论文数: 0 引用数: 0
h-index: 0
机构:
Ambit Biosci, San Diego, CA 92121 USA Ambit Biosci, San Diego, CA 92121 USA
[2]
Nagar B, 2002, CANCER RES, V62, P4236
[3]
In vitro activity of Bcr-Abl inhibitors AMN107 and BMS-354825 against clinically relevant imatinib-resistant Abl kinase domain mutants
[J].
O'Hare, T
;
Walters, DK
;
Stoffregen, EP
;
Jia, TP
;
Manley, PW
;
Mestan, J
;
Cowan-Jacob, SW
;
Lee, FY
;
Heinrich, MC
;
Deininger, MWN
;
Druker, BJ
.
CANCER RESEARCH,
2005, 65 (11)
:4500-4505

O'Hare, T
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Walters, DK
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Stoffregen, EP
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Jia, TP
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Manley, PW
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Mestan, J
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Cowan-Jacob, SW
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Lee, FY
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Heinrich, MC
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Deininger, MWN
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA

Druker, BJ
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth Sci Univ, Howard Hughes Med Inst, Inst Canc, Portland, OR 97239 USA
[4]
AMN107: Tightening the grip of imatinib
[J].
O'Hare, T
;
Walters, DK
;
Deininger, MWN
;
Druker, BJ
.
CANCER CELL,
2005, 7 (02)
:117-119

O'Hare, T
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Inst Canc, Howard Hughes Med Inst, Portland, OR 97239 USA

Walters, DK
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Inst Canc, Howard Hughes Med Inst, Portland, OR 97239 USA

Deininger, MWN
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Inst Canc, Howard Hughes Med Inst, Portland, OR 97239 USA

Druker, BJ
论文数: 0 引用数: 0
h-index: 0
机构:
Oregon Hlth & Sci Univ, Inst Canc, Howard Hughes Med Inst, Portland, OR 97239 USA Oregon Hlth & Sci Univ, Inst Canc, Howard Hughes Med Inst, Portland, OR 97239 USA
[5]
Inhibition of wild-type and mutant Bcr-Abl by AP23464, a potent ATP-based oncogenic protein kinase inhibitor: implications for CML
[J].
O'Hare, T
;
Pollock, R
;
Stoffregen, EP
;
Keats, JA
;
Abdullah, OM
;
Moseson, EM
;
Rivera, VM
;
Tang, H
;
Metcalf, CA
;
Bohacek, RS
;
Wang, YH
;
Sundaramoorthi, R
;
Shakespeare, WC
;
Dalgarno, D
;
Clackson, T
;
Sawyer, TK
;
Deininger, MW
;
Druker, BJ
.
BLOOD,
2004, 104 (08)
:2532-2539

O'Hare, T
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA

Pollock, R
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA

Stoffregen, EP
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA

Keats, JA
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA

Abdullah, OM
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA

Moseson, EM
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA

Rivera, VM
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA

Tang, H
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA

Metcalf, CA
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA

Bohacek, RS
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA

Wang, YH
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA

Sundaramoorthi, R
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA

Shakespeare, WC
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA

Dalgarno, D
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA

Clackson, T
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA

Sawyer, TK
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA

Deininger, MW
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA

Druker, BJ
论文数: 0 引用数: 0
h-index: 0
机构: Oregon Hlth & Sci Univ, Howard Hughes Med Inst, Portland, OR 97239 USA
[6]
Imatinib inhibits T-cell receptor-mediated T-cell proliferation and activation in a dose-dependent manner
[J].
Seggewiss, R
;
Loré, K
;
Greiner, E
;
Magnusson, MK
;
Price, DA
;
Douek, DC
;
Dunbar, CE
;
Wiestner, A
.
BLOOD,
2005, 105 (06)
:2473-2479

Seggewiss, R
论文数: 0 引用数: 0
h-index: 0
机构: NHLBI, Mol Hematopoiesis Sect, Hematol Branch, NIH,DHHS,Immunol Lab, Bethesda, MD 20892 USA

Loré, K
论文数: 0 引用数: 0
h-index: 0
机构: NHLBI, Mol Hematopoiesis Sect, Hematol Branch, NIH,DHHS,Immunol Lab, Bethesda, MD 20892 USA

Greiner, E
论文数: 0 引用数: 0
h-index: 0
机构: NHLBI, Mol Hematopoiesis Sect, Hematol Branch, NIH,DHHS,Immunol Lab, Bethesda, MD 20892 USA

Magnusson, MK
论文数: 0 引用数: 0
h-index: 0
机构: NHLBI, Mol Hematopoiesis Sect, Hematol Branch, NIH,DHHS,Immunol Lab, Bethesda, MD 20892 USA

Price, DA
论文数: 0 引用数: 0
h-index: 0
机构: NHLBI, Mol Hematopoiesis Sect, Hematol Branch, NIH,DHHS,Immunol Lab, Bethesda, MD 20892 USA

Douek, DC
论文数: 0 引用数: 0
h-index: 0
机构: NHLBI, Mol Hematopoiesis Sect, Hematol Branch, NIH,DHHS,Immunol Lab, Bethesda, MD 20892 USA

Dunbar, CE
论文数: 0 引用数: 0
h-index: 0
机构: NHLBI, Mol Hematopoiesis Sect, Hematol Branch, NIH,DHHS,Immunol Lab, Bethesda, MD 20892 USA

Wiestner, A
论文数: 0 引用数: 0
h-index: 0
机构: NHLBI, Mol Hematopoiesis Sect, Hematol Branch, NIH,DHHS,Immunol Lab, Bethesda, MD 20892 USA
[7]
Overriding imatinib resistance with a novel ABL kinase inhibitor
[J].
Shah, NP
;
Tran, C
;
Lee, FY
;
Chen, P
;
Norris, D
;
Sawyers, CL
.
SCIENCE,
2004, 305 (5682)
:399-401

Shah, NP
论文数: 0 引用数: 0
h-index: 0
机构: Univ Calif Los Angeles, Dept Med, Div Hematol & Oncol, Los Angeles, CA 90095 USA

Tran, C
论文数: 0 引用数: 0
h-index: 0
机构: Univ Calif Los Angeles, Dept Med, Div Hematol & Oncol, Los Angeles, CA 90095 USA

Lee, FY
论文数: 0 引用数: 0
h-index: 0
机构: Univ Calif Los Angeles, Dept Med, Div Hematol & Oncol, Los Angeles, CA 90095 USA

Chen, P
论文数: 0 引用数: 0
h-index: 0
机构: Univ Calif Los Angeles, Dept Med, Div Hematol & Oncol, Los Angeles, CA 90095 USA

Norris, D
论文数: 0 引用数: 0
h-index: 0
机构: Univ Calif Los Angeles, Dept Med, Div Hematol & Oncol, Los Angeles, CA 90095 USA

Sawyers, CL
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif Los Angeles, Dept Med, Div Hematol & Oncol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Med, Div Hematol & Oncol, Los Angeles, CA 90095 USA
[8]
Characterization of AMN107, a selective inhibitor of native and mutant Bcr-Abl
[J].
Weisberg, E
;
Manley, PW
;
Breitenstein, W
;
Brüggen, J
;
Cowan-Jacob, SW
;
Ray, A
;
Huntly, B
;
Fabbro, D
;
Fendrich, G
;
Hall-Meyers, E
;
Kung, AL
;
Mestan, J
;
Daley, GQ
;
Callahan, L
;
Catley, L
;
Cavazza, C
;
Mohammed, A
;
Neuberg, D
;
Wright, RD
;
Gilliland, DG
;
Griffin, JD
.
CANCER CELL,
2005, 7 (02)
:129-141

Weisberg, E
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Manley, PW
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Breitenstein, W
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Brüggen, J
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Cowan-Jacob, SW
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Ray, A
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Huntly, B
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Fabbro, D
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Fendrich, G
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Hall-Meyers, E
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Kung, AL
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Mestan, J
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Daley, GQ
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Callahan, L
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Catley, L
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Cavazza, C
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Mohammed, A
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Neuberg, D
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Wright, RD
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Gilliland, DG
论文数: 0 引用数: 0
h-index: 0
机构: Dana Farber Canc Inst, Boston, MA 02115 USA

Griffin, JD
论文数: 0 引用数: 0
h-index: 0
机构:
Dana Farber Canc Inst, Boston, MA 02115 USA Dana Farber Canc Inst, Boston, MA 02115 USA