Identification of ortho-amino benzamides and nicotinamides as MCHr1 antagonists

被引：22

作者：

Vasudevan, A ^{[1
]}

LaMarche, MJ

Blackburn, C

Che, JL

Luchaco-Cullis, CA

Lai, SJ

Marsilje, TH

Patane, MA

Souers, AJ

Wodka, D

Geddes, B

Chen, SM

Brodjian, S

Falls, DH

Dayton, BD

Bush, E

Brune, M

Shapiro, RD

Marsh, KC

Hernandez, LE

Sham, HL

Collins, CA

Kym, PR

机构：

[1] Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

[2] Millennium Pharmaceut Inc, Cambridge, MA 02139 USA

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 2005年 / 15卷 / 19期

关键词：

MCH; obesity; benzamides; nicotinamides; melanin concentrating hormone;

D O I：

10.1016/j.bmcl.2005.06.089

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：4174 / 4179

页数：6

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