Discovery of 6-oxo-3-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1(6H)pyridazinebutanoic acid (FK838):: A novel non-xanthine adenosine A1 receptor antagonist with potent diuretic activity

被引：107

作者：

Akahane, A ^{[1
]}

Katayama, H ^{[1
]}

Mitsunaga, T ^{[1
]}

Kato, T ^{[1
]}

Kinoshita, T ^{[1
]}

Kita, Y ^{[1
]}

Kusunoki, T ^{[1
]}

Terai, T ^{[1
]}

Yoshida, K ^{[1
]}

Shiokawa, Y ^{[1
]}

机构：

[1] Fujisawa Pharmaceut Co Ltd, Med Chem Res Labs, Yodogawa Ku, Osaka 5328514, Japan

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1999年 / 42卷 / 05期

关键词：

D O I：

10.1021/jm980671w

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：779 / 783

页数：5

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