UDP-Glucuronosyltransferase inhibitors

被引：4

作者：

Golovinsky, E ^{[1
]}

Naydenova, Z ^{[1
]}

Grancharov, K ^{[1
]}

机构：

[1] Bulgarian Acad Sci, Inst Mol Biol, BU-1113 Sofia, Bulgaria

来源：

EUROPEAN JOURNAL OF DRUG METABOLISM AND PHARMACOKINETICS | 1998年 / 23卷 / 04期

关键词：

glucuronidation; UDP-glucuronosyltransferases; detoxification pathway;

D O I：

10.1007/BF03189994

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：453 / 456

页数：4

共 32 条

[1]

Alargov DK, 1997, MONATSH CHEM, V128, P725, DOI 10.1007/BF00807604

[2] HETEROGENEITY OF HEPATIC UDP-GLUCURONOSYLTRANSFERASE ACTIVITIES - INVESTIGATIONS OF ISOENZYMES INVOLVED IN P-NITROPHENOL GLUCURONIDATION [J].

ANTOINE, B ;

BOUTIN, JA ;

SIEST, G .

COMPARATIVE BIOCHEMISTRY AND PHYSIOLOGY C-TOXICOLOGY & PHARMACOLOGY, 1993, 106 (01) :241-248

[3] CHEMICAL MODIFICATION OF HUMAN UDP-GLUCURONOSYLTRANSFERASE UGT1(ASTERISK)6 BY DIETHYL PYROCARBONATE - POSSIBLE INVOLVEMENT OF A HISTIDINE RESIDUE IN THE CATALYTIC PROCESS [J].

BATTAGLIA, E ;

PRITCHARD, M ;

OUZZINE, M ;

FOURNELGIGLEUX, S ;

RADOMINSKA, A ;

SIEST, G ;

MAGDALOU, J .

ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS, 1994, 309 (02) :266-272

[4] CHARACTERIZATION OF A NEW CLASS OF INHIBITORS OF THE RECOMBINANT HUMAN LIVER UDP-GLUCURONOSYLTRANSFERASE, UCT1-ASTERISK-6 [J].

BATTAGLIA, E ;

ELASS, A ;

DRAKE, RR ;

PAUL, P ;

TREAT, S ;

MAGDALOU, J ;

FOURNELGIGLEUX, S ;

SIEST, G ;

VERGOTEN, G ;

LESTER, R ;

RADOMINSKA, A .

BIOCHIMICA ET BIOPHYSICA ACTA-GENERAL SUBJECTS, 1995, 1243 (01) :9-14

[5] THE CHEMICAL MODIFICATION OF HUMAN LIVER UDP-GLUCURONOSYLTRANSFERASE UGT1(ASTERISK)6 REVEALS THE INVOLVEMENT OF A CARBOXYL GROUP IN CATALYSIS [J].

BATTAGLIA, E ;

SENAY, C ;

FOURNELGIGLEUX, S ;

HERBER, R ;

SIEST, G ;

MAGDALOU, J .

FEBS LETTERS, 1994, 346 (2-3) :146-150

[6]

Bock K W, 1986, Adv Exp Med Biol, V197, P171

[7]

BOCK KW, 1994, HDB EXPER PHARM, V112, P391

[8] THE MOLECULAR-BIOLOGY OF UDP-GLUCURONYLTRANSFERASES [J].

BURCHELL, B ;

JACKSON, MR ;

COARSER, RB ;

COUGHTRIE, MWH ;

HARDING, D ;

SHEPHERD, SH ;

WILSON, SM .

BIOCHEMICAL SOCIETY TRANSACTIONS, 1987, 15 (04) :581-584

[9]

CLARKE DJ, 1994, HDB EXPT PHARM, V112, P3

[10] INHIBITION OF BILIRUBIN UDPGLUCURONOSYLTRANSFERASE ACTIVITY BY TRIPHENYLACETIC ACID AND RELATED-COMPOUNDS [J].

FOURNEL, S ;

GREGOIRE, B ;

MAGDALOU, J ;

CARRE, MC ;

LAFAURIE, C ;

SIEST, G ;

CAUBERE, P .

BIOCHIMICA ET BIOPHYSICA ACTA, 1986, 883 (02) :190-196

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