Solid phase synthesis of aryl amines via palladium catalyzed amination of resin-bound aromatic bromides

被引：74

作者：

Ward, YD

Farina, V

机构：

[1] Department of Chemical Development, Boehringer Ingelheim Pharmaceut. I., Ridgefield

来源：

TETRAHEDRON LETTERS | 1996年 / 37卷 / 39期

关键词：

D O I：

10.1016/0040-4039(96)01566-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Polymer-bound aromatic bromides were found to readily undergo Pd-catalyzed amination with a number of primary and secondary alkyl- and arylamines to give, after cleavage from the support, a variety of arylamine products. Copyright (C) 1996 Elsevier Science Ltd

引用

页码：6993 / 6996

页数：4