A short and efficient synthesis of N-substituted indol-2-ones (oxindoles)

被引：10

作者：

Forbes, IT ^{[1
]}

机构：

[1] GlaxoSmithKline, Harlow CM19 5AD, Essex, England

来源：

TETRAHEDRON LETTERS | 2001年 / 42卷 / 39期

关键词：

heterocyclic compounds; indol-2-ones; oxindoles; synthesis;

D O I：

10.1016/S0040-4039(01)01413-7

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A short and high yielding process has been developed for the synthesis of N-(4-piperidinyl)-indol-2-ones. This strategy also constitutes a general route to N-substituted indol-2-ones. (C) 2001 Elsevier Science Ltd. All rights reserved.

引用

页码：6943 / 6945

页数：3

共 17 条

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